Target Details
| UniProt AC | Q9Y463 |
|---|---|
| Gene Symbol | DYRK1B |
| Protein Name | Dual specificity tyrosine-phosphorylation-regulated kinase 1B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 657
- Clinical molecules 10
- Avg pChEMBL 7.08
Associated Diseases (1)
Active Molecules (657)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QSGKPYRFWJINEH
|
9.6 | IC50 | 12 | — | |
KYOPCGIPHGGWMV
|
9.4 | IC50 | 7 | — | |
RYBNARZBIXTFJS
|
9.2 | IC50 | 9 | — | |
RYBNARZBIXTFJS
|
9.2 | IC50 | 9 | — | |
ZPXSIWLYMMFFCE
|
9.2 | IC50 | 2 | — | |
RKUKAACYUCUJEE
|
9.2 | Ki | 58 | — | |
BWRQNVDGLTUELI
|
9.0 | IC50 | 5 | — | |
DPDVVGCNUWGGRS
|
9.0 | IC50 | 10 | — | |
KHVQTEBOVFILCQ
|
9.0 | IC50 | 10 | — | |
KJCRALOGJOLXCU
|
9.0 | IC50 | 3 | — | |
KRWCFCQJKXIENS
|
9.0 | IC50 | 3 | — | |
NWMPVMMGSHXANZ
|
9.0 | Ki | 58 | — | |
PEXTWZUAIQCVBB
|
9.0 | IC50 | 3 | — | |
UBGUCDLLEIGHHP
|
9.0 | IC50 | 6 | — | |
VCTLOEWZYIGVBO
|
9.0 | IC50 | 12 | — | |
MNVPCONHWCXDES
|
9.0 | IC50 | 9 | — | |
VONVAHFLRYRXSJ
|
9.0 | IC50 | 2 | — | |
ZKGOFDAUIALGLZ
|
8.9 | IC50 | 2 | — | |
ZQVADOVUSXDTNV
|
8.8 | IC50 | 2 | — | |
RFRICXRVXVFZMF
|
8.8 | IC50 | 2 | — | |
QHTJZFWEQYRYQE
|
8.8 | IC50 | 9 | — | |
HEVBCYZPXGZFGS
|
8.7 | IC50 | 11 | — | |
BULHRWBHKAVJMT
|
8.7 | IC50 | 8 | — | |
LHQWPYOYDRVMFI
|
8.7 | Ki | 21 | — | |
QXFBTYPBHYOEMX
|
8.7 | IC50 | 9 | — | |
RJYLSCSDDDQEPD
|
8.7 | IC50 | 10 | — | |
URNZTLZSAVLTIZ
|
8.7 | Ki | 26 | — | |
HKSZLNNOFSGOKW
|
8.7 | IC50 | 408 | — | |
NMUDZNRXZXDYEQ
|
8.6 | IC50 | 9 | — | |
FUMCKNCUEAQHCV
|
8.6 | Ki | 103 | — | |
BQWWOBKMDWACGC
|
8.6 | IC50 | 8 | — | |
AVKKQBJQERVCTD
|
8.6 | IC50 | 2 | — | |
BIMZUQRAGIDOLB
|
8.5 | IC50 | 2 | — | |
QTHCAAFKVUWAFI
|
8.4 | IC50 | 23 | — | |
RDWOWHGVIKYPLI
|
8.4 | IC50 | 2 | — | |
BPNUQXPIQBZCMR
|
8.4 | Kd | 83 | Yes | |
DFMCXVONDDGQIY
|
8.4 | Ki | 66 | — | |
MHAJGINRQAEMIM
|
8.4 | IC50 | 2 | — | |
QMUKOEKTUBVPFU
|
8.4 | IC50 | 12 | — | |
YEZMGVBTPDYRPO
|
8.4 | IC50 | 8 | — | |
OTKQTETZDVGXBV
|
8.4 | IC50 | 4 | — | |
LTQMADLYBJVCSN
|
8.3 | IC50 | 2 | — | |
BGXZIBSLBRKDTP
|
8.3 | IC50 | 2 | — | |
BBCSUMURJUYILA
|
8.3 | IC50 | 10 | — | |
BDMXFIMYKGLQAL
|
8.3 | IC50 | 9 | — | |
BWNQBFHVFFZHMR
|
8.3 | IC50 | 10 | — | |
CGPYAXSYKQBYKJ
|
8.3 | IC50 | 12 | — | |
HJYHJYGXRBYDIG
|
8.3 | Ki | 23 | — | |
HKSZLNNOFSGOKW
|
8.3 | Ki | 118 | — | |
NBTJWRPKGNQBJS
|
8.3 | IC50 | 8 | — |