Target Details
| UniProt AC | Q9Y337 |
|---|---|
| Gene Symbol | KLK5 |
| Protein Name | Kallikrein-5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00089 (Trypsin) |
Summary
- Multi-target molecules 62
- Clinical molecules 0
- Avg pChEMBL 7.04
Active Molecules (62)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RDZNGZAQRWVXQR
|
9.5 | Ki | 2 | — | |
FYWPIBWNEIANCT
|
8.9 | Ki | 2 | — | |
NWAGTUQRZPXSNY
|
8.9 | IC50 | 5 | — | |
PJWRVDWTVAOOQV
|
8.7 | Ki | 7 | — | |
PBSQXKHCZCXSLI
|
8.7 | Ki | 2 | — | |
STJCUZOTQPIXIR
|
8.6 | Ki | 2 | — | |
OCOZTJLWHRDAJG
|
8.5 | IC50 | 4 | — | |
OPVLRSNIYJHUNK
|
8.5 | IC50 | 4 | — | |
WICLAAAUGCVLKH
|
8.4 | Ki | 2 | — | |
NWAGTUQRZPXSNY
|
8.3 | IC50 | 4 | — | |
NWAGTUQRZPXSNY
|
8.3 | IC50 | 6 | — | |
YENXZRUMZHNJKP
|
8.3 | IC50 | 4 | — | |
ZXLZUCADFTVDHK
|
8.3 | Ki | 3 | — | |
CZUOSFFYNSDZJT
|
8.2 | IC50 | 2 | — | |
QFJOOWSJASQPAX
|
8.2 | IC50 | 7 | — | |
LUNUFGFUBAQPEV
|
8.1 | IC50 | 4 | — | |
QMBYBZFEWIPUTA
|
8.0 | IC50 | 2 | — | |
UHZDIMFNWHQJEY
|
8.0 | IC50 | 3 | — | |
DVGJSQUHDMDLCX
|
7.9 | IC50 | 2 | — | |
PMNZGHNHIJFIAX
|
7.9 | IC50 | 2 | — | |
RXLQPJAGXHHDMC
|
7.6 | Ki | 2 | — | |
ATSZLVKWSVRBLA
|
7.6 | IC50 | 4 | — | |
FLJAMCIHLYTQCT
|
7.1 | IC50 | 4 | — | |
ZDLCAMFQMDNCSU
|
7.1 | IC50 | 2 | — | |
WUANWHWUHPZKMS
|
7.1 | IC50 | 2 | — | |
IDFLVSYGEYZZGR
|
6.8 | IC50 | 4 | — | |
MRAAINIKTLQAMC
|
6.8 | IC50 | 4 | — | |
SXIFJSHGLQMOET
|
6.8 | Ki | 3 | — | |
JTQBMTFVGGUDPN
|
6.7 | Ki | 3 | — | |
QOLOIIDNXILJRE
|
6.6 | IC50 | 4 | — | |
BIEYFOHSWAIQDF
|
6.6 | IC50 | 5 | — | |
CCNUFKYNBAVEHI
|
6.5 | IC50 | 2 | — | |
MICLUGCMNGFNIQ
|
6.5 | IC50 | 3 | — | |
VRMZLUPLYRHORK
|
6.4 | Ki | 6 | — | |
IXBWIERGNHGIDD
|
6.4 | IC50 | 2 | — | |
RBMBACCNCLXNAF
|
6.3 | IC50 | 2 | — | |
FRAFAKWXNNKJCF
|
6.3 | IC50 | 2 | — | |
KTPYVEWDDQSBAX
|
6.3 | Ki | 5 | — | |
WAZLNMJDGBJWQY
|
6.3 | IC50 | 2 | — | |
WYFUNPGYPSDKCF
|
6.3 | Ki | 3 | — | |
VKPLBOPLYIVTRL
|
6.3 | IC50 | 3 | — | |
UJHCYBGLPMMJDH
|
6.3 | IC50 | 3 | — | |
FKSBHSQGFGGOEF
|
6.2 | Ki | 4 | — | |
NYGGGQOBPHOCIJ
|
6.2 | Ki | 3 | — | |
WLGDDLRHBMVFMQ
|
6.2 | Ki | 3 | — | |
CSZFJKLNCKEZQL
|
6.2 | IC50 | 3 | — | |
RZXMQAUOJUDTRO
|
6.2 | IC50 | 2 | — | |
YLUMVCNEFHTQHD
|
6.2 | IC50 | 3 | — | |
CUGMKURPXUMGSV
|
6.1 | Ki | 4 | — | |
YJSGXHVKZSSCKV
|
6.1 | IC50 | 2 | — |