Target Details
| UniProt AC | Q9Y2U5 |
|---|---|
| Gene Symbol | MAP3K2 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00564 (PB1) PF00069 (Pkinase) |
Summary
- Multi-target molecules 36
- Clinical molecules 14
- Avg pChEMBL 6.84
KEGG Pathways (3)
Active Molecules (36)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UIARLYUEJFELEN
|
8.3 | Kd | 289 | Yes | |
XZXHXSATPCNXJR
|
8.0 | Kd | 165 | Yes | |
HKSZLNNOFSGOKW
|
7.6 | IC50 | 408 | — | |
UBPYILGKFZZVDX
|
7.5 | Kd | 130 | Yes | |
NXSJMRCTGYTSTK
|
7.4 | Kd | 200 | — | |
YRDHKIFCGOZTGD
|
7.4 | IC50 | 21 | — | |
HFNKQEVNSGCOJV
|
7.4 | Kd | 65 | — | |
OSVUGUHRKMMBSE
|
7.3 | Kd | 170 | — | |
WINHZLLDWRZWRT
|
7.2 | Kd | 201 | Yes | |
ZCCPLJOKGAACRT
|
7.2 | Kd | 599 | — | |
PIQCTGMSNWUMAF
|
7.2 | Kd | 137 | Yes | |
CTNPALGJUAXMMC
|
7.1 | Kd | 151 | — | |
KTEIFNKAUNYNJU
|
7.1 | Kd | 114 | — | |
YYLKKYCXAOBSRM
|
7.1 | Kd | 191 | — | |
GUBJNPWVIUFSTR
|
7.1 | Kd | 103 | — | |
NHHQJBCNYHBUSI
|
7.0 | Kd | 220 | — | |
QQWUGDVOUVUTOY
|
7.0 | Kd | 231 | Yes | |
BMGQWWVMWDBQGC
|
6.8 | Kd | 147 | Yes | |
FPQNRXITKTZFMF
|
6.8 | Kd | 13 | — | |
ZBNZXTGUTAYRHI
|
6.8 | Kd | 102 | Yes | |
RYYNGWLOYLRZLK
|
6.8 | Kd | 45 | — | |
APPXQUDJLJXULP
|
6.6 | IC50 | 47 | — | |
LOLPPWBBNUVNQZ
|
6.6 | Kd | 97 | Yes | |
CUIHSIWYWATEQL
|
6.5 | Kd | 61 | Yes | |
KGPGFQWBCSZGEL
|
6.5 | Kd | 59 | Yes | |
JWNPDZNEKVCWMY
|
6.3 | Kd | 57 | Yes | |
DKZYXHCYPUVGAF
|
6.3 | Kd | 112 | — | |
JOOXLOJCABQBSG
|
6.2 | Kd | 139 | — | |
VAARYSWULJUGST
|
6.2 | Kd | 119 | Yes | |
QKKIWEILHCXECO
|
6.2 | IC50 | 24 | — | |
XYASHXPUZJDWIO
|
6.2 | Kd | 7 | — | |
ZCBUQCWBWNUWSU
|
6.2 | Kd | 59 | — | |
MFAQYJIYDMLAIM
|
6.1 | Kd | 130 | Yes | |
HXNUFFCHRIWTRZ
|
6.0 | IC50 | 5 | — | |
ZZSBPGIGIUFJRA
|
6.0 | Kd | 46 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — |