Target Details
| UniProt AC | Q9Y2K2 |
|---|---|
| Gene Symbol | SIK3 |
| Protein Name | Serine/threonine-protein kinase SIK3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF23312 (UBA_SIK3) |
Summary
- Multi-target molecules 196
- Clinical molecules 8
- Avg pChEMBL 7.79
Associated Diseases (1)
Active Molecules (196)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SXMRTOWWEVQQSC
|
7.0 | IC50 | 3 | — | |
VAARYSWULJUGST
|
7.0 | Kd | 119 | Yes | |
DWTXIQAMWBBKJO
|
7.0 | IC50 | 2 | — | |
LWHNEYJBIRCBSR
|
7.0 | IC50 | 3 | — | |
DNKJWTDFPIZFNK
|
6.9 | IC50 | 3 | — | |
OASYTCDRFWTGNE
|
6.9 | IC50 | 2 | — | |
UIARLYUEJFELEN
|
6.9 | Kd | 289 | Yes | |
YFVBBRRMTKZKEK
|
6.9 | IC50 | 2 | — | |
HJHOVADSVUHROW
|
6.8 | IC50 | 3 | — | |
RIJYZTZQMRSSEU
|
6.8 | IC50 | 3 | — | |
KCUIXXONNLBRFH
|
6.8 | IC50 | 3 | — | |
NJMKEYLTIHAWEP
|
6.8 | IC50 | 3 | — | |
OYDTWNVVTPPDDO
|
6.8 | IC50 | 3 | — | |
CJGYTKZVACPSNS
|
6.7 | IC50 | 3 | — | |
UKXHMXAKNAXPBS
|
6.7 | IC50 | 3 | — | |
UKMGZRUGIXWOJQ
|
6.7 | IC50 | 3 | — | |
ZZSBPGIGIUFJRA
|
6.6 | Kd | 46 | — | |
CRLZGLXSANQWFT
|
6.6 | IC50 | 6 | — | |
QAMUWRFOZKONDU
|
6.6 | IC50 | 7 | — | |
CNFUDCYXMQHQFO
|
6.6 | IC50 | 3 | — | |
LHZJHTRTELKUDE
|
6.5 | IC50 | 2 | — | |
LXRITECWUGVGTD
|
6.5 | IC50 | 6 | — | |
PMXGPFCKENCVOL
|
6.5 | IC50 | 3 | — | |
XIAKIYQZBHRETP
|
6.5 | IC50 | 3 | — | |
DUDGRZRMJYRPNL
|
6.5 | IC50 | 2 | — | |
HJSKVVATRBELDD
|
6.5 | IC50 | 3 | — | |
RTRHXDLGBINMNM
|
6.5 | IC50 | 5 | — | |
CHPOIFDTUJGSBW
|
6.5 | IC50 | 2 | — | |
DKZYXHCYPUVGAF
|
6.5 | Kd | 112 | — | |
YFNWWNRZJGMDBR
|
6.4 | Kd | 35 | — | |
HYMHVNNHIASECU
|
6.4 | IC50 | 5 | — | |
UKBGBACORPRCGG
|
6.4 | IC50 | 17 | — | |
FNEDDGRJWXWDNZ
|
6.3 | IC50 | 5 | — | |
INSVCYRFDCTMIA
|
6.3 | IC50 | 5 | — | |
SZGFJHKSBCTFLK
|
6.3 | IC50 | 3 | — | |
UEOOSASFOHAWBP
|
6.3 | IC50 | 2 | — | |
KEGXXUKERMUSTH
|
6.2 | IC50 | 2 | — | |
TZEWBPGVTYPITP
|
6.2 | IC50 | 5 | — | |
OMZCMEYTWSXEPZ
|
6.2 | Kd | 43 | Yes | |
ZLOMEKCROOJNIA
|
6.1 | IC50 | 2 | — | |
NBCDTZGTPATHKN
|
6.1 | IC50 | 2 | — | |
NEHHEDJQRHQOOW
|
6.1 | IC50 | 5 | — | |
GMTZLHADUFDDDN
|
6.0 | IC50 | 5 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |