Target Details
| UniProt AC | Q9Y2K2 |
|---|---|
| Gene Symbol | SIK3 |
| Protein Name | Serine/threonine-protein kinase SIK3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF23312 (UBA_SIK3) |
Summary
- Multi-target molecules 196
- Clinical molecules 8
- Avg pChEMBL 7.79
Associated Diseases (1)
Active Molecules (196)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XPJFDYHVVLGXHY
|
7.9 | IC50 | 3 | — | |
CSZAJEXPQFERTK
|
7.9 | IC50 | 10 | — | |
WRPKJPATUZRQFL
|
7.9 | IC50 | 3 | — | |
QKNBRNSGPNCARD
|
7.9 | IC50 | 9 | — | |
QOOLIAIGEONMHK
|
7.9 | IC50 | 3 | — | |
VFDIZCUBJRZYFL
|
7.9 | IC50 | 3 | — | |
UWLKLAVEUJFHNV
|
7.8 | IC50 | 3 | — | |
UXTSNWGOMSEBTG
|
7.8 | IC50 | 2 | — | |
AEYQVJYAPMGHSF
|
7.8 | IC50 | 3 | — | |
IIRJOBJKMBEOMH
|
7.8 | IC50 | 3 | — | |
ZBNZXTGUTAYRHI
|
7.8 | IC50 | 102 | Yes | |
RGEJEFYGSBMYRS
|
7.8 | IC50 | 3 | — | |
VCZDFACOFNRTMG
|
7.8 | IC50 | 6 | — | |
AQXQPESYCSEOOG
|
7.7 | IC50 | 3 | — | |
IDHYGWPCQJKIOG
|
7.7 | IC50 | 3 | — | |
XCGUGTWHQADPNS
|
7.6 | IC50 | 3 | — | |
XASOHFCUIQARJT
|
7.6 | IC50 | 4 | — | |
XPSCTAWDRZNUCF
|
7.6 | IC50 | 3 | — | |
DVQJNPZTPKFTFL
|
7.6 | IC50 | 3 | — | |
CKVPYFIWJCSSSQ
|
7.6 | IC50 | 3 | — | |
IVKGWWZSELOWKX
|
7.5 | IC50 | 3 | — | |
VQINULODWGEVBB
|
7.5 | IC50 | 4 | — | |
OHQUFRHYRLCLFC
|
7.5 | IC50 | 3 | — | |
CBLISIIXOMPZFZ
|
7.5 | IC50 | 3 | — | |
RJLWSBWYWAAETQ
|
7.5 | IC50 | 3 | — | |
FWRPKNVNQNONLF
|
7.4 | IC50 | 2 | — | |
ULGBXNOOIDGVSQ
|
7.4 | IC50 | 3 | — | |
PKJTVQJCYWTEFT
|
7.4 | IC50 | 2 | — | |
SVNQOEFGBNGPSZ
|
7.4 | IC50 | 3 | — | |
PBQKEWXFKZOWAZ
|
7.4 | IC50 | 3 | — | |
IAYGCINLNONXHY
|
7.4 | Kd | 50 | — | |
JKDJAOQUTMBBQB
|
7.4 | IC50 | 5 | — | |
LZUYOYKXEXENTQ
|
7.4 | IC50 | 5 | — | |
OFIFLUFVENTCNZ
|
7.4 | IC50 | 11 | — | |
OKSHQZCQVDERIF
|
7.3 | IC50 | 3 | — | |
JPMOTSGSTDSLFB
|
7.3 | IC50 | 2 | — | |
ANQJLVHORSBOEP
|
7.3 | IC50 | 3 | — | |
PBCZSGKMGDDXIJ
|
7.2 | Kd | 68 | Yes | |
ZMNVPNNTSQXNLO
|
7.2 | IC50 | 3 | — | |
DCDKXVMMAAIMRA
|
7.2 | IC50 | 3 | — | |
WWJJXHPSYKGLJY
|
7.2 | IC50 | 2 | — | |
DFZKXFCZKLBBRG
|
7.2 | IC50 | 3 | — | |
UBPYILGKFZZVDX
|
7.2 | Kd | 130 | Yes | |
PNAUGSWMKOHDJF
|
7.2 | IC50 | 3 | — | |
JTVBXQAYBIJXRP
|
7.2 | Kd | 20 | — | |
RGUMENUIWKKDQS
|
7.1 | IC50 | 3 | — | |
WXBMZGPQDSOPBO
|
7.1 | IC50 | 2 | — | |
XSGDOSCYEQRDBE
|
7.1 | IC50 | 3 | — | |
QWACVNYZRLANPQ
|
7.1 | IC50 | 2 | — | |
BMGQWWVMWDBQGC
|
7.0 | Kd | 147 | Yes |