Target Details
| UniProt AC | Q9Y2K2 |
|---|---|
| Gene Symbol | SIK3 |
| Protein Name | Serine/threonine-protein kinase SIK3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF23312 (UBA_SIK3) |
Summary
- Multi-target molecules 196
- Clinical molecules 8
- Avg pChEMBL 7.79
Associated Diseases (1)
Active Molecules (196)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XELNNUJRQXCODY
|
8.5 | IC50 | 3 | — | |
ZXYITDGKYOBFAO
|
8.5 | IC50 | 3 | — | |
HWSYLCVSNZMWCP
|
8.5 | IC50 | 3 | — | |
BIYKGGOFJOFQIZ
|
8.5 | IC50 | 3 | — | |
JXJARIRMZQINMV
|
8.4 | IC50 | 3 | — | |
WKZOFECSVXLTOB
|
8.4 | IC50 | 3 | — | |
GRPZYURNHYVZBO
|
8.4 | IC50 | 3 | — | |
UNBNKYSPLOMIOY
|
8.4 | IC50 | 7 | — | |
NELFAFAXIZFQJB
|
8.4 | IC50 | 3 | — | |
NQANXDMJOUTFBB
|
8.4 | IC50 | 3 | — | |
FCJGMZMSVIAAJU
|
8.4 | IC50 | 9 | — | |
MGMOBQWMSWOTLL
|
8.4 | IC50 | 3 | — | |
RXHXLESLBWUVQS
|
8.4 | IC50 | 3 | — | |
SGMHSWUFNYQVBA
|
8.4 | IC50 | 9 | — | |
HRKJFKJZUNJKNU
|
8.4 | IC50 | 10 | — | |
JDNFAAUUFUBZKC
|
8.4 | IC50 | 3 | — | |
QYFGVVMJUHWKNB
|
8.3 | IC50 | 3 | — | |
AQXQPESYCSEOOG
|
8.3 | IC50 | 3 | — | |
INDWAJWLSOYKGH
|
8.3 | IC50 | 3 | — | |
CAJPKOHOPAWXRV
|
8.3 | IC50 | 3 | — | |
QBSNPDJXAMBWIZ
|
8.3 | IC50 | 3 | — | |
MXJMJNRCJKHFPP
|
8.3 | IC50 | 10 | — | |
AWVUPXUQWGNTHF
|
8.3 | IC50 | 3 | — | |
FQZGWTSGSBKLBT
|
8.2 | IC50 | 3 | — | |
JPVJPXAQFGYJDI
|
8.2 | IC50 | 3 | — | |
YPGZOVPNRGMYIT
|
8.2 | IC50 | 3 | — | |
AZCVMDQKOWCQAG
|
8.2 | IC50 | 3 | — | |
LZCGMQZFMKDCSR
|
8.2 | IC50 | 2 | — | |
SVJBHQPXESBDEQ
|
8.2 | IC50 | 9 | — | |
WEHOIIGXTMKVRG
|
8.2 | IC50 | 3 | — | |
WWTRFWLRGARRAD
|
8.2 | IC50 | 10 | — | |
GTSDNTZRPRBMTP
|
8.2 | IC50 | 3 | — | |
JVBRZBKYIRZVJE
|
8.1 | IC50 | 3 | — | |
HSYDEPQAUCZNGP
|
8.1 | IC50 | 3 | — | |
RPDJXKWOAHHTBX
|
8.1 | IC50 | 3 | — | |
SIICZZZVCXGXGX
|
8.1 | IC50 | 3 | — | |
XOZORSAAPNHXFP
|
8.1 | IC50 | 3 | — | |
MYYIXDJCLRMEBI
|
8.1 | IC50 | 3 | — | |
NXSJMRCTGYTSTK
|
8.0 | Kd | 200 | — | |
UEQMHAFWQDRPMU
|
8.0 | IC50 | 3 | — | |
WCLYSPWUHSZWOR
|
8.0 | IC50 | 3 | — | |
BYKVUESQXQHBEP
|
8.0 | IC50 | 7 | — | |
PJFVPKCPIJSWQT
|
8.0 | IC50 | 3 | — | |
QIUASFSNWYMDFS
|
8.0 | Kd | 5 | — | |
ZGIZZXHFELWYTH
|
8.0 | IC50 | 3 | — | |
OMDTWHBLOYOZGL
|
7.9 | IC50 | 3 | — | |
UGMDEPACJFWQTK
|
7.9 | IC50 | 3 | — | |
YHKXOSIWOVIDSP
|
7.9 | IC50 | 3 | — | |
NCQKIKYQHVNIMN
|
7.9 | IC50 | 2 | — | |
XCGUGTWHQADPNS
|
7.9 | IC50 | 3 | — |