Target Details
| UniProt AC | Q9Y2K2 |
|---|---|
| Gene Symbol | SIK3 |
| Protein Name | Serine/threonine-protein kinase SIK3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF23312 (UBA_SIK3) |
Summary
- Multi-target molecules 196
- Clinical molecules 8
- Avg pChEMBL 7.79
Associated Diseases (1)
Active Molecules (196)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KDPXVKRYHKSBPY
|
9.4 | IC50 | 3 | — | |
FPNPNYBQZUNHGQ
|
9.2 | IC50 | 3 | — | |
PFTXFNSHFZLJNT
|
9.2 | IC50 | 17 | — | |
FGLQSISJARINNB
|
9.2 | IC50 | 3 | — | |
HOKRUYIIDRQYFK
|
9.1 | IC50 | 3 | — | |
DYMFNPBLDKXKJA
|
9.1 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
9.0 | IC50 | 408 | — | |
VNWAWEZKWMFEJY
|
9.0 | IC50 | 6 | — | |
WDNAXOPVZIEECR
|
9.0 | IC50 | 11 | — | |
WXCYMIOQVROELY
|
9.0 | IC50 | 3 | — | |
ARXQRVVEKOEUEV
|
9.0 | IC50 | 3 | — | |
XHPICGSLCSAZKX
|
9.0 | IC50 | 3 | — | |
YMSJZKSIBUPNHN
|
9.0 | IC50 | 3 | — | |
VCQQIZTUIHARTH
|
8.9 | IC50 | 3 | — | |
LTQKUGJNXFIXKC
|
8.9 | IC50 | 3 | — | |
VATIVDMNNPRBCN
|
8.9 | IC50 | 3 | — | |
VOYZWDQJVPQGCO
|
8.9 | IC50 | 9 | — | |
ZMAJVXKEVISHMQ
|
8.9 | IC50 | 9 | — | |
YCOQHBLWDSAZRB
|
8.9 | IC50 | 3 | — | |
SHMKAHZOTDZUIN
|
8.8 | IC50 | 3 | — | |
XGEBOBAOVSOQCV
|
8.8 | IC50 | 10 | — | |
QVUYJTWSZWCKHP
|
8.8 | IC50 | 3 | — | |
AWLHPMOLJAWKDL
|
8.8 | IC50 | 3 | — | |
HSQLWSUNRMTGGO
|
8.8 | IC50 | 3 | — | |
YOWQNRVRQMOXAT
|
8.8 | IC50 | 3 | — | |
DEJPFOVGKKDPLD
|
8.8 | IC50 | 3 | — | |
KAUKMJZXRPFGAB
|
8.8 | IC50 | 3 | — | |
KNOCCCXGASNIAF
|
8.8 | IC50 | 3 | — | |
KZVDQIXBUFBWLM
|
8.8 | IC50 | 3 | — | |
MMGVIQXQPXLHQK
|
8.8 | IC50 | 3 | — | |
MXNBWDNCIZQCIL
|
8.8 | IC50 | 3 | — | |
YATIMLFNGFQTCA
|
8.8 | IC50 | 3 | — | |
INXQKXZSUNICKV
|
8.7 | IC50 | 3 | — | |
WMCHGBLGKMZDJD
|
8.7 | IC50 | 3 | — | |
BHFWGYATBPONNI
|
8.7 | IC50 | 3 | — | |
BIYKGGOFJOFQIZ
|
8.7 | IC50 | 3 | — | |
DYNHJHQFHQTFTP
|
8.7 | Kd | 38 | — | |
CFNFPVIKPAPVOV
|
8.7 | IC50 | 3 | — | |
PZFORNOVSGDEAS
|
8.7 | IC50 | 3 | — | |
CAWABSRZIMATJO
|
8.7 | IC50 | 9 | — | |
NDNNIKHUOLIORS
|
8.7 | IC50 | 3 | — | |
RZXPVLRGCBTJSU
|
8.7 | IC50 | 3 | — | |
JWADUJSXPDSTOX
|
8.7 | IC50 | 3 | — | |
LYSXGFLZKDKZDF
|
8.6 | IC50 | 3 | — | |
OLULSQINUASNMI
|
8.6 | IC50 | 3 | — | |
XVNZURGXHLXJIR
|
8.6 | IC50 | 3 | — | |
BQKJBKRZMBOHNT
|
8.6 | IC50 | 3 | — | |
UARVSLPFGRKWQN
|
8.5 | IC50 | 11 | — | |
AQSSMEORRLJZLU
|
8.5 | Kd | 34 | Yes | |
MBBASLHNWYZIRZ
|
8.5 | IC50 | 3 | — |