Target Details
| UniProt AC | Q9Y2I7 |
|---|---|
| Gene Symbol | PIKFYVE |
| Protein Name | 1-phosphatidylinositol 3-phosphate 5-kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00118 (Cpn60_TCP1) PF00610 (DEP) PF01363 (FYVE) PF01504 (PIP5K) |
Summary
- Multi-target molecules 6
- Clinical molecules 0
- Avg pChEMBL 7.73
KEGG Pathways (6)
Associated Diseases (1)
Active Molecules (6)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CUVPKJMJOAUYEQ
|
9.3 | Kd | 2 | — | |
DGLFSNZWRYADFC
|
8.7 | IC50 | 12 | — | |
DORZPJWJOBMQKC
|
8.4 | IC50 | 9 | — | |
MJJJRRMQCUUKEO
|
7.4 | IC50 | 3 | — | |
LHIXDFRNBOEPTF
|
6.6 | IC50 | 3 | — | |
XCOSAQGGGZDYJN
|
6.0 | Kd | 11 | — |