Target Details
| UniProt AC | Q9Y2H9 |
|---|---|
| Gene Symbol | MAST1 |
| Protein Name | Microtubule-associated serine/threonine-protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08926 (DUF1908) PF17820 (PDZ_6) PF00069 (Pkinase) |
Summary
- Multi-target molecules 11
- Clinical molecules 5
- Avg pChEMBL 6.6
Associated Diseases (1)
Active Molecules (11)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UIARLYUEJFELEN
|
7.7 | Kd | 289 | Yes | |
PIQCTGMSNWUMAF
|
7.4 | Kd | 137 | Yes | |
HKSZLNNOFSGOKW
|
6.8 | Kd | 408 | — | |
BMGQWWVMWDBQGC
|
6.7 | Kd | 147 | Yes | |
WINHZLLDWRZWRT
|
6.7 | Kd | 201 | Yes | |
CTNPALGJUAXMMC
|
6.5 | Kd | 151 | — | |
UBPYILGKFZZVDX
|
6.5 | Kd | 130 | Yes | |
HFNKQEVNSGCOJV
|
6.3 | Kd | 65 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |