Target Details
| UniProt AC | Q9Y271 |
|---|---|
| Gene Symbol | CYSLTR1 |
| Protein Name | Cysteinyl leukotriene receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 386
- Clinical molecules 1
- Avg pChEMBL 7.62
KEGG Pathways (2)
Active Molecules (386)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RDEBUULLBLDEFT
|
6.3 | IC50 | 2 | — | |
XPHYAOVCSFEMLP
|
6.3 | IC50 | 2 | — | |
JRLOEMCOOZSCQP
|
6.3 | IC50 | 4 | Yes | |
JVCPEXLEPXEVOW
|
6.3 | Kd | 2 | — | |
UCWVNGPPUUVQRU
|
6.3 | Ki | 2 | — | |
RZENAZZCHMPRHI
|
6.2 | IC50 | 2 | — | |
IYWIRJBMFCOWHN
|
6.2 | Ki | 2 | — | |
LGFNWYHWAVUQBZ
|
6.2 | IC50 | 2 | — | |
WZLAUXKXTLNMDW
|
6.2 | IC50 | 2 | — | |
FWLOXRGJZILONQ
|
6.2 | Kd | 2 | — | |
HJVFWIQQGMVLMN
|
6.2 | IC50 | 2 | — | |
WOOGNRDKJXUFCT
|
6.2 | IC50 | 2 | — | |
CCKAUHCWAKYDHV
|
6.2 | IC50 | 2 | — | |
PNLVUVAWZGCJHS
|
6.2 | Ki | 2 | — | |
PZMVLVOWRMBYQH
|
6.2 | IC50 | 2 | — | |
QXRHBPIFLPGMQO
|
6.2 | Ki | 2 | — | |
QLCZDHMXLNJXHS
|
6.2 | Ki | 2 | — | |
GHYJLDJJOTYUQB
|
6.2 | IC50 | 2 | — | |
RLCNRWRACMSPHG
|
6.1 | Kd | 2 | — | |
NQJREPQHJNEAAW
|
6.1 | IC50 | 2 | — | |
MARJKKBMAPXHAK
|
6.1 | IC50 | 2 | — | |
MWYHLEQJTQJHSS
|
6.1 | Ki | 2 | — | |
MYSHIWFTLJUGST
|
6.1 | IC50 | 2 | — | |
MLVOIYGTXJJNAP
|
6.1 | Kd | 2 | — | |
OMZOJDVVRPSXSI
|
6.1 | IC50 | 2 | — | |
WWQFMCKPIBAFRI
|
6.1 | Ki | 2 | — | |
LRGJBPUUPFFZRB
|
6.0 | Ki | 2 | — | |
WHPYNUNVBQASGT
|
6.0 | Kd | 2 | — | |
FITIWWKKLYDKFT
|
6.0 | Ki | 2 | — | |
IPUAPZIXPYVKRA
|
6.0 | IC50 | 2 | — | |
KOMGKDHFTYYZRF
|
6.0 | IC50 | 2 | — | |
MSZAYVGTGJPGBY
|
6.0 | IC50 | 2 | — | |
OZESMWJKGNPCBZ
|
6.0 | Ki | 2 | — | |
RLUZFDUUXQPYEI
|
6.0 | IC50 | 2 | — | |
XFZHNLAPVOHWLM
|
6.0 | IC50 | 2 | — | |
ZDJMZZUUHCSCKL
|
6.0 | IC50 | 2 | — |