Target Details
| UniProt AC | Q9Y271 |
|---|---|
| Gene Symbol | CYSLTR1 |
| Protein Name | Cysteinyl leukotriene receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 386
- Clinical molecules 1
- Avg pChEMBL 7.62
KEGG Pathways (2)
Active Molecules (386)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OKPACELMVBBRER
|
6.7 | IC50 | 2 | — | |
QSEWBONWOPSITJ
|
6.7 | IC50 | 2 | — | |
LEONVQOXNVQAHC
|
6.6 | Kd | 2 | — | |
HUNHHUAGWDAVDL
|
6.6 | IC50 | 2 | — | |
VLPMDPRPICKPJS
|
6.6 | Kd | 2 | — | |
HPDCVSUTOBCBFF
|
6.6 | Ki | 2 | — | |
FKMWHFNAFDBNRL
|
6.6 | IC50 | 2 | — | |
JZKKFABLTBZDCS
|
6.6 | IC50 | 2 | — | |
LAURNBCWALNAEO
|
6.6 | IC50 | 2 | — | |
GTHFHADQTUOWAA
|
6.6 | IC50 | 2 | — | |
IIHHSWYDPCUBAX
|
6.5 | IC50 | 2 | — | |
OYKPWSZSBLRRPL
|
6.5 | IC50 | 11 | — | |
PNCHHOQSFSFTLA
|
6.5 | Ki | 2 | — | |
QJLULXIBQDCMAN
|
6.5 | IC50 | 2 | — | |
CEWRLAYRDVWJEE
|
6.5 | IC50 | 2 | — | |
LLQPCGSXHFGKFV
|
6.5 | IC50 | 2 | — | |
PULYGNHSSUPCKL
|
6.5 | IC50 | 2 | — | |
UBXFQYMXDODOLD
|
6.5 | Ki | 2 | — | |
WEWBWUMLTYFQDQ
|
6.5 | IC50 | 2 | — | |
HAWPNKMQRDDAER
|
6.5 | Kd | 2 | — | |
UIEQEUSTJLJAMM
|
6.5 | IC50 | 2 | — | |
QAFXJLKSSNVBDG
|
6.5 | IC50 | 2 | — | |
RHGRRGBOSFJRBE
|
6.5 | IC50 | 2 | — | |
JXDQWYZHYXKUMS
|
6.5 | Kd | 2 | — | |
FOECKIWHCOYYFL
|
6.4 | IC50 | 4 | — | |
HGBUQTOGNIRVHU
|
6.4 | IC50 | 2 | — | |
BDUWLAJHXQHPPO
|
6.4 | Ki | 2 | — | |
BVCCOBUJFKURIJ
|
6.4 | IC50 | 2 | — | |
CNXDZCJGGWJKPO
|
6.4 | IC50 | 2 | — | |
GYVDSWAEYLAXKJ
|
6.4 | IC50 | 2 | — | |
JZFFHOCNJWSHKJ
|
6.4 | Kd | 2 | — | |
YNHQJUJPBNEXHQ
|
6.4 | Ki | 2 | — | |
CZJYWNTYOQKSBJ
|
6.4 | IC50 | 2 | — | |
JXVXKIYLTSMUSV
|
6.4 | IC50 | 2 | — | |
KGNOOMFHDAFWMR
|
6.4 | IC50 | 2 | — | |
FYTRQOCBJGGXJC
|
6.4 | Ki | 2 | — | |
ZEWCLTWIGFQTFS
|
6.4 | Ki | 2 | — | |
PKJINWOACFYDQN
|
6.4 | IC50 | 2 | — | |
TUKZDRAVAURZLG
|
6.4 | Ki | 2 | — | |
DOJFGABESYVMQD
|
6.3 | Kd | 2 | — | |
PEDBVGXUGSZQBG
|
6.3 | Ki | 2 | — | |
POSBEAIEWFUXQK
|
6.3 | IC50 | 2 | — | |
NHNMQZGEZGQBBW
|
6.3 | Ki | 2 | — | |
SQQYQKRQLZICSQ
|
6.3 | IC50 | 2 | — | |
KAIRIRDEGZVHEP
|
6.3 | IC50 | 2 | — | |
USNXDIGYHYCXRZ
|
6.3 | Ki | 2 | — | |
WNCBAUIHJHOYFZ
|
6.3 | IC50 | 2 | — | |
CWQKHAHDLWFTAV
|
6.3 | IC50 | 2 | — | |
JNEGTBPWGUPOJQ
|
6.3 | IC50 | 2 | — | |
OBKYYCSRBOOXHT
|
6.3 | IC50 | 2 | — |