Target Details
| UniProt AC | Q9Y271 |
|---|---|
| Gene Symbol | CYSLTR1 |
| Protein Name | Cysteinyl leukotriene receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 386
- Clinical molecules 1
- Avg pChEMBL 7.62
KEGG Pathways (2)
Active Molecules (386)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VZKVRBRBVFYTPT
|
7.0 | IC50 | 2 | — | |
YNRLZKIONIAXNM
|
7.0 | IC50 | 2 | — | |
YPUUTNJQPHSGDA
|
7.0 | IC50 | 2 | — | |
UKKDVBPLHLWOJP
|
7.0 | IC50 | 2 | — | |
VZXSJDNSOOGZCG
|
7.0 | IC50 | 2 | — | |
GEPCPHZJFQZONY
|
7.0 | Ki | 2 | — | |
BYTUMFJCBKNJKZ
|
6.9 | IC50 | 2 | — | |
JRLYDKCKUUVXLK
|
6.9 | IC50 | 2 | — | |
MGYZMMFPQHHKTJ
|
6.9 | IC50 | 2 | — | |
VCPKGFRGDDVSMP
|
6.9 | IC50 | 2 | — | |
AJWHKNGJIRLMHT
|
6.9 | IC50 | 2 | — | |
JSWCCMIJFXNTGD
|
6.9 | Ki | 2 | — | |
SQQTUVOFASOKGW
|
6.9 | IC50 | 2 | — | |
BWDRKHWOKWDREA
|
6.8 | IC50 | 2 | — | |
DHVCRZJQBSNOHZ
|
6.8 | Ki | 2 | — | |
FGXYVESYEYBLLQ
|
6.8 | Ki | 2 | — | |
FOTHBOISNKWERK
|
6.8 | IC50 | 2 | — | |
IQRQDDCMOXNYHM
|
6.8 | Kd | 2 | — | |
PWEJTHONIDHCLI
|
6.8 | IC50 | 2 | — | |
YNJADCKFFBHTQO
|
6.8 | IC50 | 2 | — | |
QOPFKXVYVLMQQY
|
6.8 | IC50 | 2 | — | |
GEZVDUJVSIHSRL
|
6.8 | Ki | 2 | — | |
FLVULROWBMBEMN
|
6.8 | IC50 | 2 | — | |
HFGIVBJHCTYWRO
|
6.8 | IC50 | 2 | — | |
CEZOAWAOXBVCPM
|
6.8 | Ki | 2 | — | |
LMQBMWHHGVZWMR
|
6.8 | IC50 | 2 | — | |
WLYVFAOLHPVBSD
|
6.8 | IC50 | 2 | — | |
HYTBIVFDTLBKQS
|
6.8 | IC50 | 2 | — | |
KKKANLNLSLPJEX
|
6.8 | Kd | 2 | — | |
JHKJAWIANIFNJV
|
6.7 | IC50 | 2 | — | |
FLDYGLHLJSKGRL
|
6.7 | Kd | 2 | — | |
XXVSAUUGDHWSDC
|
6.7 | Ki | 2 | — | |
MJDLJMHJJYEQFO
|
6.7 | IC50 | 2 | — | |
PQQBUGBOBWUDPV
|
6.7 | Kd | 2 | — | |
ASTFJODCVHJWJI
|
6.7 | IC50 | 2 | — | |
FZYPHWZZKVKYCO
|
6.7 | IC50 | 2 | — | |
HNPGZXUDAMBXBD
|
6.7 | IC50 | 2 | — | |
KNLAAKYVFWRDNZ
|
6.7 | IC50 | 2 | — | |
PFNMDMFQJFQOLA
|
6.7 | IC50 | 2 | — | |
RHBHCSGKNNYBCZ
|
6.7 | IC50 | 2 | — | |
WYXYQZDZCYKRKJ
|
6.7 | IC50 | 2 | — | |
XYDDTGWBQPOONX
|
6.7 | Kd | 2 | — | |
YSTYSNAKWCYTAV
|
6.7 | IC50 | 2 | — | |
HSGFYFLPTLCPMD
|
6.7 | Kd | 2 | — | |
LMSOJQRZAUJDRM
|
6.7 | Kd | 2 | — | |
FIJKMECDVUAIRF
|
6.7 | IC50 | 2 | — | |
JHGLTDMWVRBYTB
|
6.7 | Kd | 2 | — | |
SRAYUFAGOZRLIA
|
6.7 | IC50 | 2 | — | |
VBWDQBKEADPPMZ
|
6.7 | Kd | 2 | — | |
RMHXCEHCZLOYMR
|
6.7 | IC50 | 2 | — |