Target Details
| UniProt AC | Q9Y271 |
|---|---|
| Gene Symbol | CYSLTR1 |
| Protein Name | Cysteinyl leukotriene receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 386
- Clinical molecules 1
- Avg pChEMBL 7.62
KEGG Pathways (2)
Active Molecules (386)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YTYIEGFQGGDPOC
|
7.9 | IC50 | 2 | — | |
KEAPEQBCDVILQF
|
7.9 | IC50 | 2 | — | |
UQJBBYJBUQUDNA
|
7.9 | IC50 | 2 | — | |
IWEUQSCUBLQJOC
|
7.8 | IC50 | 2 | — | |
MONJECLHXLONHX
|
7.8 | Ki | 2 | — | |
RQGVZKQWFKFPHB
|
7.8 | IC50 | 2 | — | |
RYSLZFOZDSIPHK
|
7.8 | Ki | 2 | — | |
AQNPOVSLJSQEIU
|
7.8 | Ki | 2 | — | |
OMZSXMJYCZJLNG
|
7.8 | IC50 | 2 | — | |
XNLJGFSXSWPVCV
|
7.8 | IC50 | 2 | — | |
CZKMNFXLXQKWLQ
|
7.8 | IC50 | 2 | — | |
XXQDVVUJZWUKJS
|
7.8 | IC50 | 2 | — | |
CCNFJZLJCWVIGY
|
7.8 | IC50 | 2 | — | |
YMCYOKUMKYELQN
|
7.8 | Ki | 2 | — | |
MULRRAQIDXPIJO
|
7.7 | IC50 | 2 | — | |
CLXLXWOOKSJSED
|
7.7 | IC50 | 2 | — | |
OQMSTTQHFRKDFE
|
7.7 | Ki | 2 | — | |
LMIDOCUHJVWTNG
|
7.7 | IC50 | 2 | — | |
PICBIHJXRQGHJG
|
7.7 | IC50 | 2 | — | |
XYJIAOBZIHRGLX
|
7.7 | IC50 | 2 | — | |
YBNVSQIAVPPCOR
|
7.7 | IC50 | 2 | — | |
YKYNDIGNKWVGIO
|
7.7 | Ki | 2 | — | |
OXRKVTBERXJUQW
|
7.7 | IC50 | 2 | — | |
POTRPJSXTYBGAD
|
7.7 | Ki | 2 | — | |
SILSWXVHSFRLCM
|
7.7 | Kd | 2 | — | |
QLCYDOOHNFRQMA
|
7.7 | Ki | 2 | — | |
XFDWMOIFWMJDPH
|
7.7 | IC50 | 2 | — | |
CPTPCKPMEIITER
|
7.6 | IC50 | 2 | — | |
JVBGKXGXUZCESP
|
7.6 | Ki | 2 | — | |
KQXMBUWEISAGDL
|
7.6 | IC50 | 2 | — | |
OBGPJXBAEABRDU
|
7.6 | IC50 | 2 | — | |
FJOGJBNZYBZBSZ
|
7.6 | Ki | 2 | — | |
ITUHVJQASQRAST
|
7.6 | IC50 | 2 | — | |
OVHFPPKAUNIZRJ
|
7.6 | Kd | 2 | — | |
SZDFJWULJMPHIK
|
7.6 | IC50 | 2 | — | |
UGLUMKDNDDXQAB
|
7.6 | IC50 | 2 | — | |
XCUTWBWDDQNSEQ
|
7.6 | Ki | 2 | — | |
URIMHZHMIDRURZ
|
7.6 | IC50 | 2 | — | |
HXALHRWESQWBPV
|
7.6 | Kd | 2 | — | |
IXJCHVMUTFCRBH
|
7.6 | Ki | 2 | — | |
TUKZDRAVAURZLG
|
7.6 | Ki | 2 | — | |
UZESQRCECKSIRG
|
7.5 | IC50 | 2 | — | |
FYQQKKWEXPVKTH
|
7.5 | Ki | 2 | — | |
PBGVAFUTEIUHFM
|
7.5 | Ki | 2 | — | |
XGDMPCXGTASNNX
|
7.5 | IC50 | 2 | — | |
IRNLQQDWCBJNCF
|
7.5 | IC50 | 2 | — | |
ROKIOTZMRLYACP
|
7.5 | IC50 | 2 | — | |
VATIUDIQNXIBGY
|
7.5 | IC50 | 2 | — | |
GABZVHZCIWHURT
|
7.5 | Ki | 2 | — | |
LSWRNJJFSREPHH
|
7.5 | IC50 | 2 | — |