Target Details
| UniProt AC | Q9Y271 |
|---|---|
| Gene Symbol | CYSLTR1 |
| Protein Name | Cysteinyl leukotriene receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 386
- Clinical molecules 1
- Avg pChEMBL 7.62
KEGG Pathways (2)
Active Molecules (386)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JITXEOCUBFNDSU
|
8.5 | IC50 | 2 | — | |
ICYLDMBMBLPBFJ
|
8.4 | IC50 | 2 | — | |
VFXGMPUTFGTYBV
|
8.4 | IC50 | 2 | — | |
ZAVSTDHOBGBUAC
|
8.4 | IC50 | 2 | — | |
SUDSSIJBZOKIID
|
8.4 | IC50 | 2 | — | |
JKUHAVTVPYKANI
|
8.3 | IC50 | 2 | — | |
BPSQDOLGQQVYNF
|
8.3 | IC50 | 2 | — | |
JOVCMJZWLGTFAU
|
8.3 | IC50 | 2 | — | |
PMIIRTOUWKTUSF
|
8.3 | IC50 | 2 | — | |
PTQNWRHPFTVLJE
|
8.3 | IC50 | 2 | — | |
NWOCFLOMBOQAIR
|
8.3 | IC50 | 2 | — | |
ZPNLVCLQVZRJJJ
|
8.3 | IC50 | 2 | — | |
DTAIREAVRYTIHY
|
8.2 | Ki | 2 | — | |
FOERRCYLHSJHPT
|
8.2 | IC50 | 2 | — | |
DJGUHTJMEJTYSH
|
8.2 | IC50 | 2 | — | |
UAZVAVXMYLMNGU
|
8.2 | Kd | 2 | — | |
KMDMEBAGSHHFKW
|
8.2 | IC50 | 2 | — | |
QNKLTIIDWGBTQS
|
8.2 | IC50 | 2 | — | |
FZWBSDKVGGBWAW
|
8.2 | Ki | 2 | — | |
GYKCTIBPYOPSIN
|
8.2 | IC50 | 2 | — | |
PQBWZIFOPYSMTQ
|
8.1 | IC50 | 2 | — | |
HOXJOAWSVADHMC
|
8.1 | IC50 | 2 | — | |
QQZLHBYIEUHFBH
|
8.1 | IC50 | 2 | — | |
HEPNHAYVEMEOKU
|
8.1 | IC50 | 2 | — | |
IEISNEYLXZRMDU
|
8.1 | Ki | 2 | — | |
ALCIWBPDUXMXBZ
|
8.1 | IC50 | 2 | — | |
AIANCPCQGZTGKM
|
8.1 | IC50 | 2 | — | |
KEPHPBWTZIPAJX
|
8.1 | IC50 | 2 | — | |
PHPYDISUCJTNJT
|
8.1 | IC50 | 2 | — | |
CZEPGSHEVIBKCM
|
8.0 | IC50 | 2 | — | |
JTTSKYBQFRJIPS
|
8.0 | IC50 | 2 | — | |
LFXZDWFKMMTVNE
|
8.0 | IC50 | 2 | — | |
LJEADJFDJNIWOM
|
8.0 | Ki | 2 | — | |
OKLGLROKXFUYEI
|
8.0 | IC50 | 2 | — | |
PZIFPMYXXCAOCC
|
8.0 | Ki | 2 | — | |
AXUZQJFHDNNPFG
|
8.0 | Ki | 3 | — | |
BSBGMXWCCNLNRH
|
8.0 | Ki | 2 | — | |
CCNFJZLJCWVIGY
|
8.0 | IC50 | 2 | — | |
MINFQFJDELKPIC
|
8.0 | IC50 | 2 | — | |
NXMVUMPPOABACO
|
8.0 | IC50 | 2 | — | |
XLJUOMJRMGBMGV
|
8.0 | IC50 | 2 | — | |
APFHYXSUIMWOIF
|
7.9 | IC50 | 2 | — | |
GDNFOLXYEODGCP
|
7.9 | IC50 | 2 | — | |
POSUQRXFCPPYHP
|
7.9 | Ki | 2 | — | |
DBUXZZTVAHXKSD
|
7.9 | IC50 | 2 | — | |
GFXMMBLNWKLBAM
|
7.9 | Kd | 2 | — | |
GSZWFDBWUNJPJB
|
7.9 | IC50 | 2 | — | |
KIRCILKHNTZTFS
|
7.9 | IC50 | 2 | — | |
LQAREGHVTIHGAM
|
7.9 | IC50 | 2 | — | |
QADPCENSPWQNNH
|
7.9 | IC50 | 2 | — |