Target Details
| UniProt AC | Q9Y271 |
|---|---|
| Gene Symbol | CYSLTR1 |
| Protein Name | Cysteinyl leukotriene receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 386
- Clinical molecules 1
- Avg pChEMBL 7.62
KEGG Pathways (2)
Active Molecules (386)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JRMPZUJDLLDLKO
|
9.1 | IC50 | 2 | — | |
CKLRKPMEGUXCIX
|
9.1 | IC50 | 2 | — | |
YTYZMTWLPBHKJN
|
9.1 | IC50 | 2 | — | |
CCQQISILGFBECU
|
9.1 | IC50 | 2 | — | |
PNHUIGYHBQXQAN
|
9.1 | IC50 | 2 | — | |
IGUFQFBMEPZVOT
|
9.0 | IC50 | 2 | — | |
KBYYEZWFRXRCIU
|
9.0 | IC50 | 2 | — | |
NBQKINXMPLXUET
|
9.0 | IC50 | 2 | — | |
UKCJWCGWHOCIIK
|
9.0 | IC50 | 2 | — | |
XBNBASSLEBZZPC
|
9.0 | IC50 | 2 | — | |
NGIBWHCRTISQMK
|
9.0 | IC50 | 2 | — | |
WMVFGKBJSVBHEK
|
9.0 | IC50 | 2 | — | |
XRJAXAKIACIPIF
|
9.0 | IC50 | 2 | — | |
XWWWRDGIDIASEO
|
8.9 | IC50 | 2 | — | |
NUUXRXDZKMLTMN
|
8.9 | Kd | 2 | — | |
DKJWFOPJQMKRJT
|
8.9 | IC50 | 2 | — | |
AOFPEKPLQQABJA
|
8.9 | IC50 | 2 | — | |
NWPVERDHSASZCG
|
8.9 | IC50 | 2 | — | |
OQHBFPBWKNCKGR
|
8.8 | Ki | 2 | — | |
XKPRBHVTNOLIBA
|
8.8 | IC50 | 2 | — | |
XXFIWZPRMVGKBH
|
8.8 | IC50 | 2 | — | |
BALDTNWRBBIKOY
|
8.8 | IC50 | 2 | — | |
CJJZKNPQCCVQGX
|
8.8 | IC50 | 2 | — | |
NTBXOFAJPMVAEU
|
8.8 | IC50 | 2 | — | |
VAAUGWQPDBPVHS
|
8.8 | IC50 | 2 | — | |
WMNXRPRPIGXCDK
|
8.8 | IC50 | 2 | — | |
SILHYVDKGHXGBL
|
8.8 | IC50 | 2 | — | |
TUENNGAJMWSHCB
|
8.8 | IC50 | 2 | — | |
YEEZWCHGZNKEEK
|
8.7 | IC50 | 5 | — | |
DSUJZPQYEUITAA
|
8.7 | Kd | 2 | — | |
FKGPTFPCZZCYKN
|
8.7 | IC50 | 2 | — | |
KBBBPRAKKDDMRH
|
8.7 | IC50 | 2 | — | |
NRQPBWTZSUTFDI
|
8.7 | IC50 | 2 | — | |
OQMSTTQHFRKDFE
|
8.7 | Ki | 2 | — | |
WVQDGTOQBZZIAO
|
8.7 | IC50 | 2 | — | |
SPRSDGHQROEUPI
|
8.6 | IC50 | 2 | — | |
XLYKIVOUGYCXDI
|
8.6 | IC50 | 2 | — | |
VMSCZLCBWYPUAI
|
8.6 | IC50 | 2 | — | |
IBDAOFPNZMUFAK
|
8.6 | IC50 | 2 | — | |
ZPIFAXSOEFMHAL
|
8.6 | IC50 | 2 | — | |
PJVNGFRHENPVNP
|
8.6 | IC50 | 2 | — | |
CTNCLMQKMHDOHK
|
8.5 | IC50 | 2 | — | |
KIUKUOYAZCSXNU
|
8.5 | IC50 | 2 | — | |
JELDFLOBXROBFH
|
8.5 | Ki | 2 | — | |
NVUKVULDQXPOLM
|
8.5 | IC50 | 2 | — | |
PWYWVEHZMASOIG
|
8.5 | Ki | 2 | — | |
UKECUOUDZYOQPY
|
8.5 | IC50 | 2 | — | |
YVRKZBMFZRCTDJ
|
8.5 | IC50 | 2 | — | |
SVEIXTCDRMVORE
|
8.5 | IC50 | 2 | — | |
AWYSEGZBFYYQQL
|
8.5 | IC50 | 2 | — |