Target Details
| UniProt AC | Q9Y251 |
|---|---|
| Gene Symbol | HPSE |
| Protein Name | Heparanase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF03662 (Glyco_hydro_79n) |
Summary
- Multi-target molecules 35
- Clinical molecules 0
- Avg pChEMBL 7.2
KEGG Pathways (3)
Active Molecules (35)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ABJDIWGVGOYYNM
|
8.4 | Ki | 3 | — | |
WSRYCXXKENQCDY
|
8.3 | Ki | 3 | — | |
MVGUXRGOSPSVTI
|
8.2 | Ki | 3 | — | |
AENWAPDCFRFKIF
|
8.2 | Ki | 3 | — | |
LNUFLCYMSVYYNW
|
8.2 | Ki | 3 | — | |
IPWXMKVZKOEZQH
|
8.2 | Ki | 3 | — | |
MIKHBYRVCGYIJG
|
8.1 | Ki | 3 | — | |
MTFFLFAICAKCHG
|
8.1 | Ki | 3 | — | |
CVHJGGCCDHKCBI
|
8.0 | Ki | 3 | — | |
VENGQIUBROEMGG
|
8.0 | Ki | 3 | — | |
GQXXCBAPTBXUNH
|
8.0 | Ki | 3 | — | |
OBNDKQCXTGZBFN
|
8.0 | Ki | 3 | — | |
ODJIBJUXPSKWRB
|
7.8 | Ki | 3 | — | |
UAEGWXRHPSXZEC
|
7.7 | Ki | 3 | — | |
ZHPDNFVCUVRXEV
|
7.7 | Ki | 2 | — | |
SJTQHYMLYPZEID
|
7.5 | Ki | 2 | — | |
IPOGMIXXMPIMID
|
7.4 | Kd | 4 | — | |
IFJPUFGQBDHFEF
|
6.6 | Kd | 4 | — | |
WLVBREMNPAKRNM
|
6.6 | Kd | 4 | — | |
ZMQXKELQMWICHL
|
6.6 | Kd | 3 | — | |
LCULSEGLGJAWDH
|
6.5 | Kd | 3 | — | |
UTAMZBVYPTVJDJ
|
6.5 | Kd | 4 | — | |
SWIQMDRPSXMESL
|
6.5 | Kd | 4 | — | |
ZCBJBKMXIXCLCT
|
6.5 | Kd | 4 | — | |
FKGOJYRHEWGRBI
|
6.5 | Kd | 4 | — | |
OFKKNRXXSSSMMU
|
6.5 | Kd | 4 | — | |
BFTCQYFPGMEWCA
|
6.5 | Kd | 4 | — | |
NVPBRXOUVIHLNN
|
6.5 | Kd | 4 | — | |
REQUDOPWXGQSHG
|
6.4 | Kd | 4 | — | |
SKQGENOFFSMNGR
|
6.4 | Kd | 4 | — | |
PSNHLUHUOQZMFM
|
6.4 | Kd | 4 | — | |
QVWJDZKITFFVCA
|
6.4 | IC50 | 2 | — | |
FCQUVPLCJSCNPK
|
6.3 | IC50 | 2 | — | |
NLMIWFMNJNSVBJ
|
6.2 | Kd | 4 | — | |
RBWDOUOLUKRISD
|
6.2 | Kd | 4 | — |