Target Details
| UniProt AC | Q9Y233 |
|---|---|
| Gene Symbol | PDE10A |
| Protein Name | cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01590 (GAF) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 348
- Clinical molecules 0
- Avg pChEMBL 7.63
KEGG Pathways (4)
Associated Diseases (2)
Active Molecules (348)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QRWHTFXNHZLJAL
|
6.4 | IC50 | 5 | — | |
WYICFGQGWWSBFA
|
6.4 | IC50 | 2 | — | |
NJMQPZWDQHNHOI
|
6.3 | IC50 | 2 | — | |
UIOIRPSCJNRZQH
|
6.3 | IC50 | 2 | — | |
VTRFAKGBUDJZNQ
|
6.3 | IC50 | 2 | — | |
DNDNLFXKQSTINI
|
6.3 | IC50 | 4 | — | |
CNSTWFCIWOBGDU
|
6.3 | IC50 | 6 | — | |
GDQXJMLXEYSICD
|
6.3 | IC50 | 6 | — | |
HVYWAAXJQNGKRV
|
6.3 | Ki | 3 | — | |
NBSFRDYQPJRINF
|
6.3 | IC50 | 2 | — | |
DXFHYPOGHCSSLE
|
6.3 | IC50 | 2 | — | |
HNISNVVBMZPQOH
|
6.3 | IC50 | 2 | — | |
IJWBPPMGHOPKJH
|
6.3 | IC50 | 2 | — | |
OZPFEONEPSBCQR
|
6.3 | IC50 | 2 | — | |
XWKUFRPLYDBTSK
|
6.3 | IC50 | 2 | — | |
PUOYLPXSDKMJBT
|
6.2 | IC50 | 2 | — | |
MZLGPWMELUQSRS
|
6.2 | IC50 | 3 | — | |
RILYOAAADBABEY
|
6.2 | IC50 | 2 | — | |
XWMJQGHYURZPMZ
|
6.2 | IC50 | 2 | — | |
GDSDBZHPAZMARE
|
6.2 | IC50 | 2 | — | |
FCIZPPJLBOLIRV
|
6.2 | IC50 | 5 | — | |
BAZNAGLQESOABE
|
6.2 | IC50 | 2 | — | |
JISGWKBRIFXTKG
|
6.2 | IC50 | 2 | — | |
XOXQBNCDSZCOJT
|
6.2 | IC50 | 2 | — | |
FOZFBBKUKXGMND
|
6.2 | IC50 | 6 | — | |
FBZARNOHVPPHSV
|
6.1 | IC50 | 2 | — | |
JQWUZRQDRJVXDJ
|
6.1 | IC50 | 3 | — | |
DHCZQKVLJXPKFJ
|
6.1 | IC50 | 2 | — | |
BJUKJODXDRHWBI
|
6.1 | IC50 | 2 | — | |
KOVUQUXRMIAWMX
|
6.1 | IC50 | 3 | — | |
DZAUSKKPHXFGNN
|
6.1 | IC50 | 6 | — | |
MNFCPURQCIBMOM
|
6.1 | IC50 | 2 | — | |
SECKRCOLJRRGGV
|
6.1 | IC50 | 16 | — | |
LFBHHJIXURBMIW
|
6.1 | IC50 | 2 | — | |
QEZMDSAIBIOKNZ
|
6.1 | IC50 | 2 | — | |
RIOWALIOYFJZSC
|
6.0 | IC50 | 2 | — | |
YMOWLMZNUJCNMI
|
6.0 | IC50 | 2 | — | |
OIDQRHGTWLIKKZ
|
6.0 | IC50 | 5 | — | |
GPPXOIFHTCJBAO
|
6.0 | IC50 | 2 | — | |
RGHSXVXSIDRFBH
|
6.0 | IC50 | 2 | — | |
MXIRJRIBGCCKEU
|
6.0 | IC50 | 2 | — | |
MYTWOYABQDJPSU
|
6.0 | IC50 | 2 | — | |
DGTJUXLZPAKEDG
|
6.0 | IC50 | 2 | — | |
IMUWQOKSBPPDFX
|
6.0 | IC50 | 2 | — | |
IZEKFCXSFNUWAM
|
6.0 | Ki | 19 | — | |
JITUOVWOCIXEEZ
|
6.0 | IC50 | 23 | — | |
LLFCUYYOIIWTAK
|
6.0 | IC50 | 2 | — | |
UYGQNCZCLDANJQ
|
6.0 | IC50 | 2 | — |