Target Details
| UniProt AC | Q9Y233 |
|---|---|
| Gene Symbol | PDE10A |
| Protein Name | cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01590 (GAF) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 348
- Clinical molecules 0
- Avg pChEMBL 7.63
KEGG Pathways (4)
Associated Diseases (2)
Active Molecules (348)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZUGQSSCMJHOUMY
|
6.8 | IC50 | 4 | — | |
DEATUVSNGIWELQ
|
6.8 | IC50 | 2 | — | |
GPICUZIEERHFCU
|
6.8 | IC50 | 2 | — | |
KDIUPJCSYMXVFK
|
6.8 | IC50 | 2 | — | |
XZXHAZRYGADTJG
|
6.8 | Ki | 3 | — | |
IVUDESFQCKKLHE
|
6.8 | IC50 | 2 | — | |
VCBMUUABISIFFN
|
6.7 | IC50 | 2 | — | |
HGUAETYOXGYETL
|
6.7 | IC50 | 2 | — | |
IEQOYZRPRRCNMO
|
6.7 | Ki | 2 | — | |
RMDSNENKGQYVPN
|
6.7 | IC50 | 2 | — | |
SCCFCNSNLMFVCF
|
6.7 | IC50 | 2 | — | |
HMHCDRWOANPTIA
|
6.7 | IC50 | 2 | — | |
PLHMFMNGOAPGBB
|
6.7 | Ki | 3 | — | |
MUCWSKZPOCCFHR
|
6.7 | IC50 | 2 | — | |
DGOKEVUAUHBVCV
|
6.7 | IC50 | 2 | — | |
QOWBGPIVWUACNE
|
6.6 | IC50 | 2 | — | |
RORWDTCBTBGWNA
|
6.6 | IC50 | 7 | — | |
IWQJRWQPBCCRGZ
|
6.6 | IC50 | 8 | — | |
NTJSCTYPHZJWMH
|
6.6 | IC50 | 2 | — | |
OVSHRJGAYOZGQR
|
6.6 | IC50 | 8 | — | |
PHAZQDYQAKMELH
|
6.6 | IC50 | 2 | — | |
QHAIBIZBWSNNOQ
|
6.6 | IC50 | 2 | — | |
DJVBNZMSHDWOSI
|
6.5 | IC50 | 2 | — | |
DPCKYZFJQHZXHN
|
6.5 | IC50 | 2 | — | |
UAMPLPXKYMJMRA
|
6.5 | IC50 | 2 | — | |
BEIVLBDHGFLMCE
|
6.5 | IC50 | 2 | — | |
GHSXQEOEHMFLKT
|
6.5 | IC50 | 2 | — | |
JODONPFHDDVTRP
|
6.5 | IC50 | 2 | — | |
QBYKGPDSZZURMK
|
6.5 | IC50 | 2 | — | |
QPOIPSGKGQTIEH
|
6.5 | IC50 | 2 | — | |
ZSDUWOZPBUPSHE
|
6.5 | IC50 | 2 | — | |
CLRZKWDDCHPPFI
|
6.5 | IC50 | 2 | — | |
XPZGQEQXHLMAGF
|
6.5 | IC50 | 2 | — | |
GUZDCVDZFPPFHH
|
6.5 | IC50 | 2 | — | |
AGNJYCZMGAQTHM
|
6.5 | IC50 | 2 | — | |
GWNXVUOBUDPUMJ
|
6.5 | IC50 | 2 | — | |
OFZGCAMFVYIIHV
|
6.5 | IC50 | 24 | — | |
PWYZKRUNIMYNFO
|
6.5 | IC50 | 2 | — | |
RBCRJQPVIVEDMI
|
6.5 | IC50 | 2 | — | |
NMOJAFKVPFGPMJ
|
6.5 | IC50 | 2 | — | |
ZUKHTEAHHSGTQU
|
6.5 | IC50 | 2 | — | |
NYTIKOBWCYNNCW
|
6.4 | IC50 | 2 | — | |
GTUZKDHSJKUJHG
|
6.4 | IC50 | 2 | — | |
NFDRPYVQPHIFFA
|
6.4 | IC50 | 2 | — | |
OOMWWAGKPLNKNM
|
6.4 | IC50 | 2 | — | |
HQUIEUONYYTHEW
|
6.4 | IC50 | 5 | — | |
WLARZYDGOHEBCG
|
6.4 | IC50 | 2 | — | |
JTROLECZHRVLFM
|
6.4 | IC50 | 10 | — | |
OFBDYPOKLBUABM
|
6.4 | IC50 | 2 | — | |
SQYNPZYBHGTSOY
|
6.4 | IC50 | 5 | — |