Target Details
| UniProt AC | Q9Y233 |
|---|---|
| Gene Symbol | PDE10A |
| Protein Name | cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01590 (GAF) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 348
- Clinical molecules 0
- Avg pChEMBL 7.63
KEGG Pathways (4)
Associated Diseases (2)
Active Molecules (348)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VNWKVRSLWCIUCC
|
7.3 | IC50 | 7 | — | |
MXWNMGSRQFJJAP
|
7.3 | IC50 | 2 | — | |
XLZOIIVTFPXQAK
|
7.3 | IC50 | 2 | — | |
IARWHEJRGFEBLP
|
7.3 | IC50 | 2 | — | |
LAUDMPJASNSMFC
|
7.3 | IC50 | 2 | — | |
RPLZXBUKXSYWDQ
|
7.3 | IC50 | 10 | — | |
VFFZRVLFFCXMEW
|
7.3 | Ki | 7 | — | |
DUXDVVOHXOPNKD
|
7.3 | Ki | 3 | — | |
OKZITNMVZCTKEZ
|
7.3 | IC50 | 2 | — | |
PUECNZWNMCIENI
|
7.3 | IC50 | 2 | — | |
GWIPZYBIMCNGCR
|
7.2 | Ki | 3 | — | |
PRDXEDQLSDAYKR
|
7.2 | IC50 | 2 | — | |
MHBOLMRBSQYNJE
|
7.2 | IC50 | 2 | — | |
RYZQUDKQJHQEFH
|
7.2 | IC50 | 2 | — | |
UNKPGLPMRWHIHZ
|
7.2 | IC50 | 2 | — | |
LEVUGPXUDZVOIL
|
7.2 | Ki | 3 | — | |
VSCSTNZWXBTXLI
|
7.2 | Ki | 3 | — | |
XRRVDIXCRUNODY
|
7.2 | IC50 | 2 | — | |
SDYQZLQJADODFL
|
7.2 | Ki | 7 | — | |
NRDAQXSEPMKYFE
|
7.1 | IC50 | 2 | — | |
CTBSIWZADWNGPL
|
7.1 | IC50 | 2 | — | |
MCCMQVOHAUUTCR
|
7.1 | IC50 | 2 | — | |
RRPOHESBIMXJJV
|
7.1 | IC50 | 2 | — | |
ZPXNETLHTOLAQO
|
7.1 | IC50 | 2 | — | |
XMDHYKYUFULFTG
|
7.1 | IC50 | 2 | — | |
VQYHPUHKYSSEOB
|
7.1 | IC50 | 5 | — | |
VJJRKPCCZNXZKA
|
7.1 | IC50 | 2 | — | |
DJXXFFAIELEXJW
|
7.0 | IC50 | 2 | — | |
OFLQGOAFVYORIF
|
7.0 | IC50 | 2 | — | |
WKGHKBGIEMZFHT
|
7.0 | IC50 | 2 | — | |
WUQPRMFKNDQDDT
|
7.0 | Ki | 3 | — | |
LRBQTFPUUPFJQW
|
7.0 | IC50 | 2 | — | |
FDQFJBXHRLSJAL
|
7.0 | Ki | 2 | — | |
ZNDBGOQQHAKYTD
|
7.0 | IC50 | 2 | — | |
BGXBOFDQKJHQGK
|
7.0 | IC50 | 2 | — | |
RYTQEZNQUVMBSA
|
7.0 | IC50 | 2 | — | |
UGVVCZOCYNUTOE
|
7.0 | IC50 | 2 | — | |
IWUVRKQUYQTUCZ
|
7.0 | Ki | 3 | — | |
CMRKQOBLHMEDQF
|
6.9 | IC50 | 2 | — | |
RPRWDECRYAMVMA
|
6.9 | IC50 | 2 | — | |
BAPYHGMPJNBMLE
|
6.9 | IC50 | 2 | — | |
LKJQBYPVUKVMQU
|
6.9 | IC50 | 2 | — | |
CEPHQHUNHIGGLV
|
6.9 | Ki | 3 | — | |
OVZFILNQGLNPAO
|
6.9 | IC50 | 2 | — | |
BMHAOZUJNXVLNI
|
6.9 | IC50 | 2 | — | |
BJMBBXFCGSCMCV
|
6.9 | IC50 | 3 | — | |
CMJKEYGSFOILJO
|
6.9 | Ki | 3 | — | |
RCUCFFJDNMXZAV
|
6.9 | Ki | 7 | — | |
YZYLQUFRZHTRQI
|
6.9 | IC50 | 2 | — | |
VQEVGOOIMFPGBB
|
6.9 | Ki | 3 | — |