Target Details
| UniProt AC | Q9Y233 |
|---|---|
| Gene Symbol | PDE10A |
| Protein Name | cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01590 (GAF) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 348
- Clinical molecules 0
- Avg pChEMBL 7.63
KEGG Pathways (4)
Associated Diseases (2)
Active Molecules (348)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YCWMLVXTEBFVHL
|
7.8 | Ki | 3 | — | |
MQPLDEMSGYODSF
|
7.7 | Ki | 3 | — | |
QLMQWJMFOGJTAL
|
7.7 | IC50 | 2 | — | |
ZVHAIWYVZBCKIO
|
7.7 | Ki | 3 | — | |
WQCSFVSIVBVUFZ
|
7.7 | Ki | 3 | — | |
CBPBGAAUJILPTQ
|
7.7 | IC50 | 2 | — | |
KTVOIZSPBSYWIC
|
7.7 | IC50 | 2 | — | |
OIOIOFDJPMGWSE
|
7.7 | IC50 | 2 | — | |
OQHKHTONZCAETM
|
7.7 | Ki | 2 | — | |
SOMBFHHGZYERAW
|
7.7 | IC50 | 3 | — | |
CEDPQOAAUSEXPN
|
7.7 | IC50 | 2 | — | |
SZMWOWPIZBQHLK
|
7.7 | Ki | 2 | — | |
HLHJPSPCRBIQQL
|
7.7 | IC50 | 2 | — | |
OOKPOAVUCNJJLK
|
7.7 | IC50 | 2 | — | |
OXQHUSMIVFYSJK
|
7.6 | IC50 | 2 | — | |
VSPLHWROJCSRNJ
|
7.6 | IC50 | 2 | — | |
XAQBODRJFGSLRC
|
7.6 | IC50 | 2 | — | |
JHNQIJOFPJQWJX
|
7.6 | IC50 | 2 | — | |
DQPTWPRWYXHDGO
|
7.6 | IC50 | 2 | — | |
MMJDOWOZKGXPBB
|
7.6 | IC50 | 2 | — | |
TUBLFDLSEINHAR
|
7.6 | Ki | 2 | — | |
WIWOBGNIVSRLMD
|
7.6 | Ki | 2 | — | |
ZTBPCVNOICVBPF
|
7.6 | Ki | 2 | — | |
AQRCAEFOEVCQPT
|
7.5 | IC50 | 2 | — | |
DKAIIUQWPLZTEM
|
7.5 | Ki | 2 | — | |
LPZCANRRYYLKAQ
|
7.5 | IC50 | 2 | — | |
QINZPNYWORORJH
|
7.5 | IC50 | 2 | — | |
QRQLCTXXSWRKOM
|
7.5 | Ki | 2 | — | |
HXWSGMZHUJKHOE
|
7.5 | IC50 | 2 | — | |
LZRGPVBUCASWQB
|
7.5 | IC50 | 2 | — | |
MKNKYIBULNNKQR
|
7.5 | IC50 | 2 | — | |
PQLTZXWSOPPUKC
|
7.5 | Ki | 2 | — | |
QVUMIQCLVPRUBJ
|
7.5 | IC50 | 2 | — | |
YDOZLNHCYOKRDQ
|
7.5 | IC50 | 2 | — | |
YHJHPCMSWXKLIU
|
7.5 | IC50 | 2 | — | |
GFIAXSKRRKHJBD
|
7.5 | Ki | 2 | — | |
WREDJOGPAYNGKD
|
7.4 | IC50 | 2 | — | |
XQYZDYMELSJDRZ
|
7.4 | IC50 | 4 | — | |
AXNJNPPDLFAOFG
|
7.4 | Ki | 2 | — | |
ASJRPPJEYHNNET
|
7.4 | IC50 | 2 | — | |
CIHGAHYOOKAOLL
|
7.4 | IC50 | 2 | — | |
KNIOZKBZHBPMPJ
|
7.4 | IC50 | 2 | — | |
XNYYCWIPILCSBL
|
7.4 | IC50 | 2 | — | |
IBGPYPKZYDRSAJ
|
7.4 | IC50 | 2 | — | |
INRSGLNDAUKKFJ
|
7.4 | IC50 | 2 | — | |
NDASMCYFWCEUSG
|
7.4 | Ki | 3 | — | |
WEXUJYQUJXVVRL
|
7.4 | IC50 | 2 | — | |
ZDOSWEGEZXKDLA
|
7.3 | IC50 | 2 | — | |
BIAGKVLTBOXOIO
|
7.3 | IC50 | 2 | — | |
OSQYQSYCOOIVGE
|
7.3 | IC50 | 2 | — |