Target Details
| UniProt AC | Q9Y233 |
|---|---|
| Gene Symbol | PDE10A |
| Protein Name | cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01590 (GAF) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 348
- Clinical molecules 0
- Avg pChEMBL 7.63
KEGG Pathways (4)
Associated Diseases (2)
Active Molecules (348)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QBLWGJRSTWQUGT
|
8.2 | IC50 | 8 | — | |
AAJCENMHNPMXLK
|
8.1 | IC50 | 2 | — | |
GWIFWBBQCOIOLL
|
8.1 | IC50 | 2 | — | |
LDBXDKOHGLAACS
|
8.1 | IC50 | 2 | — | |
WYHTXPAKFZNNJB
|
8.1 | IC50 | 4 | — | |
HZQYJFKDDWTULI
|
8.1 | IC50 | 2 | — | |
MVPONTPZYKDJPY
|
8.1 | IC50 | 3 | — | |
RMKFHXBPLKSLMZ
|
8.1 | IC50 | 3 | — | |
SQZHNYUQGYHEOQ
|
8.1 | IC50 | 2 | — | |
LXNUCQLVMSHVOF
|
8.1 | IC50 | 2 | — | |
PEQLYWXDQWUMMO
|
8.1 | Ki | 2 | — | |
WNHVXXRODSTYDN
|
8.1 | IC50 | 2 | — | |
NEAVXSYDFFCBNJ
|
8.1 | IC50 | 3 | — | |
VIQYGEOSRSOQKW
|
8.1 | Ki | 3 | — | |
MGVXODADYYKJPQ
|
8.1 | IC50 | 2 | — | |
BLODSLLFPYATAO
|
8.0 | IC50 | 2 | — | |
OVFNIEPLLFYLGK
|
8.0 | IC50 | 2 | — | |
HLUWBLAYMFWHOF
|
8.0 | IC50 | 8 | — | |
CYERGDRLLOCHQC
|
8.0 | Ki | 3 | — | |
DHCUFPIRHGVRLF
|
8.0 | IC50 | 2 | — | |
IHOKJRCFBXFQQC
|
8.0 | IC50 | 2 | — | |
VAYNYSLGOOSRMO
|
8.0 | IC50 | 2 | — | |
WBJAKXOIBNITGN
|
8.0 | IC50 | 2 | — | |
YLDDMTIJXUXGIW
|
8.0 | IC50 | 2 | — | |
YNADXFWEXJTQSZ
|
8.0 | IC50 | 4 | — | |
QAKWVFQSSVUOOT
|
8.0 | IC50 | 2 | — | |
KFGXEXAVKVJZCX
|
7.9 | Ki | 3 | — | |
PRIVQPMFDOJWFJ
|
7.9 | Ki | 2 | — | |
RLWDDGNDSFIKAI
|
7.9 | Ki | 3 | — | |
RNLNRXGCWGOQMW
|
7.9 | Ki | 7 | — | |
UPTQSRGSSJRBKJ
|
7.9 | Ki | 3 | — | |
WLBFHVBWNVZOKE
|
7.9 | IC50 | 2 | — | |
BEQMIMLEDMHHBZ
|
7.9 | IC50 | 2 | — | |
HXCMWAGIKQHTTN
|
7.9 | IC50 | 2 | — | |
MWLFLDJUMFIHDC
|
7.9 | IC50 | 2 | — | |
YNHQXCDMFQRWLP
|
7.9 | IC50 | 2 | — | |
ZMWZDEJCMAPCAG
|
7.9 | IC50 | 2 | — | |
CIKOPVDFPXGTDP
|
7.9 | IC50 | 8 | — | |
DNMZGQJGUUMZHN
|
7.9 | IC50 | 2 | — | |
UEHYTJCPYRCAPM
|
7.9 | IC50 | 8 | — | |
DGISDXJWSURSPJ
|
7.9 | IC50 | 2 | — | |
PFHNYXFZVYZXGX
|
7.8 | IC50 | 2 | — | |
KVQOOHOAWKKRAQ
|
7.8 | IC50 | 2 | — | |
VCYNWUHOQVCKIZ
|
7.8 | IC50 | 2 | — | |
AGPUZKAVMNQKCV
|
7.8 | IC50 | 2 | — | |
LPDZZRZIMYOFQN
|
7.8 | IC50 | 2 | — | |
SCPBTWMZLCCZTO
|
7.8 | IC50 | 2 | — | |
GZMAIQUXVJGBDN
|
7.8 | IC50 | 2 | — | |
UBIIFKJMNRPNMT
|
7.8 | IC50 | 3 | — | |
XUCXEJHCWUEFBU
|
7.8 | IC50 | 2 | — |