Target Details
| UniProt AC | Q9Y233 |
|---|---|
| Gene Symbol | PDE10A |
| Protein Name | cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01590 (GAF) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 348
- Clinical molecules 0
- Avg pChEMBL 7.63
KEGG Pathways (4)
Associated Diseases (2)
Active Molecules (348)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MLJILDFMLRVIKN
|
8.8 | IC50 | 2 | — | |
PMOGXWRUBZRFGT
|
8.8 | Ki | 3 | — | |
WTHIWWQIRPIFLQ
|
8.8 | IC50 | 8 | — | |
XFCSSYSGGAIHKK
|
8.8 | IC50 | 2 | — | |
OOOKPENMJKOYJM
|
8.8 | IC50 | 2 | — | |
SMBDWRLHTIVDJR
|
8.8 | IC50 | 2 | — | |
YWQRGPGREXLLMW
|
8.8 | IC50 | 2 | — | |
GMVMJTOBEXWBGG
|
8.8 | IC50 | 2 | — | |
VWEVGRMBISXBDM
|
8.8 | IC50 | 2 | — | |
LPLOWECFLAFSLK
|
8.7 | IC50 | 2 | — | |
OADIRORPIWSRQU
|
8.7 | IC50 | 3 | — | |
SUMRAEKZGBJUHZ
|
8.7 | IC50 | 2 | — | |
IYYROKXNJZBPGJ
|
8.7 | IC50 | 2 | — | |
OJPMZYKWMBETBC
|
8.7 | IC50 | 2 | — | |
VOUAUMKVLOMARH
|
8.7 | Ki | 2 | — | |
WFSLPYROCMIATC
|
8.7 | IC50 | 2 | — | |
YAGLFTIBFQFZJH
|
8.7 | Ki | 2 | — | |
CYGLUSHREFGBMF
|
8.7 | IC50 | 2 | — | |
FIUCLBJMUGCQTF
|
8.6 | IC50 | 8 | — | |
DWSJBSVHCVJEDX
|
8.6 | IC50 | 6 | — | |
FNTGJJLOKISHIS
|
8.6 | IC50 | 3 | — | |
DYFFQXLHZJUSTD
|
8.5 | IC50 | 2 | — | |
OTKDXQUDAQCPRM
|
8.5 | IC50 | 2 | — | |
ULKIELHDMWBCFZ
|
8.5 | IC50 | 6 | — | |
ZYOUAODGFIHHBS
|
8.5 | IC50 | 2 | — | |
SIGZFMSWUAQLPX
|
8.5 | IC50 | 2 | — | |
CWJZCMLRNFECBA
|
8.4 | IC50 | 2 | — | |
FHILGPQALCJBPN
|
8.4 | IC50 | 3 | — | |
FDVCQTUMHBUUBK
|
8.4 | Ki | 2 | — | |
KNPRYLFUIRHVFZ
|
8.4 | IC50 | 2 | — | |
LZYLOUZRUVTOJN
|
8.4 | IC50 | 2 | — | |
SXFYSRMCZRZBKE
|
8.4 | IC50 | 2 | — | |
KKGNLHFXELBTHO
|
8.4 | IC50 | 2 | — | |
MSAZJEUMUSIUHQ
|
8.4 | IC50 | 2 | — | |
BTYONSNIAIDRLB
|
8.4 | Ki | 3 | — | |
FOCSRCJRUICCOO
|
8.4 | IC50 | 2 | — | |
AQCSZBJZPWCJBX
|
8.3 | IC50 | 2 | — | |
IZGYMSVTXLRXSF
|
8.3 | IC50 | 2 | — | |
VGNZBEMBWAXVEK
|
8.3 | IC50 | 3 | — | |
BJZXDRJWGJFCMN
|
8.3 | IC50 | 2 | — | |
MIATWQLLYKUWRD
|
8.3 | IC50 | 8 | — | |
NASINOLFIIRYNU
|
8.3 | IC50 | 2 | — | |
XCTJCGBYOUBBCH
|
8.3 | IC50 | 2 | — | |
GEVPWAZNJXIORL
|
8.2 | IC50 | 2 | — | |
FUIPSYTUCLZFMN
|
8.2 | IC50 | 2 | — | |
OYQMVYLFCJQBFJ
|
8.2 | IC50 | 2 | — | |
IZIINKYFYLUKNA
|
8.2 | IC50 | 2 | — | |
YQQZBBVGXNRWDB
|
8.2 | Ki | 2 | — | |
FMHQKWMVSBVGPC
|
8.2 | IC50 | 2 | — | |
YWLVSEKLYMROTP
|
8.2 | IC50 | 4 | — |