Target Details
| UniProt AC | Q9Y233 |
|---|---|
| Gene Symbol | PDE10A |
| Protein Name | cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01590 (GAF) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 348
- Clinical molecules 0
- Avg pChEMBL 7.63
KEGG Pathways (4)
Associated Diseases (2)
Active Molecules (348)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DWLPNEAIQATTGD
|
11.1 | Ki | 3 | — | |
JOKHDDDMDHGDNV
|
10.4 | IC50 | 4 | — | |
HDPASTSLENKNQX
|
10.3 | IC50 | 2 | — | |
ZHLLRTLCOXWEIS
|
10.2 | IC50 | 2 | — | |
PUJFXPWIBOJQHB
|
10.2 | IC50 | 12 | — | |
SPTLTOMHDUZGDO
|
10.2 | Ki | 2 | — | |
RFLZKIMBCYCKIA
|
10.1 | IC50 | 2 | — | |
HMJXSCNBHAGAML
|
10.0 | IC50 | 2 | — | |
UJLHNYPXKZJKLV
|
10.0 | IC50 | 24 | — | |
JOJOWCOCCMULDU
|
10.0 | IC50 | 5 | — | |
RMWWNYKNAPEPNW
|
9.9 | IC50 | 4 | — | |
UWMFXMIHNIGVKF
|
9.9 | IC50 | 2 | — | |
KXCOKRBRUWINCT
|
9.9 | IC50 | 24 | — | |
UBWSOHYIVVIMQK
|
9.8 | IC50 | 2 | — | |
KPFFPWNKWSYQFT
|
9.8 | IC50 | 24 | — | |
CPFAZCJKWPHSEL
|
9.7 | Ki | 2 | — | |
IIKAIGZIYWPSLV
|
9.7 | IC50 | 2 | — | |
GOBQSCBEINUNFL
|
9.6 | IC50 | 24 | — | |
UWKQLVTVYOHHBY
|
9.6 | IC50 | 2 | — | |
ZXGQTWGCVTUQHJ
|
9.6 | IC50 | 8 | — | |
KPCVLACNFAKGBK
|
9.5 | Ki | 2 | — | |
AFCWMWBOATWMJV
|
9.5 | IC50 | 24 | — | |
DKSKKVAOIPURFT
|
9.5 | IC50 | 24 | — | |
SSDLYRZGRCSRIU
|
9.5 | IC50 | 2 | — | |
ZTLRRRPDWBCINJ
|
9.5 | IC50 | 4 | — | |
VVBTTWHJRZWRPW
|
9.5 | IC50 | 2 | — | |
MTYKIQDYUJLUDE
|
9.4 | Ki | 2 | — | |
VEYWHNZHTOXBLT
|
9.4 | IC50 | 3 | — | |
HBIJATLZLNIQGM
|
9.3 | IC50 | 2 | — | |
CUJLFJITXUBBRJ
|
9.3 | IC50 | 2 | — | |
ASGYMMSFTYPPJZ
|
9.3 | IC50 | 2 | — | |
WVFZLLHYILMVBO
|
9.2 | Ki | 7 | — | |
QQHJRLKSCSRMEM
|
9.2 | IC50 | 2 | — | |
JGRMMBRYUDVUAI
|
9.2 | IC50 | 3 | — | |
SCPJKGGAIWBYON
|
9.2 | IC50 | 2 | — | |
WLMFGIKOAOYYJI
|
9.2 | IC50 | 2 | — | |
ACOOVXAIHUBKJQ
|
9.1 | IC50 | 2 | — | |
JWFAMJCCIUWJGA
|
9.1 | IC50 | 2 | — | |
LUIFKRLOZBLHEV
|
9.1 | IC50 | 2 | — | |
WDRWBLDUZZTZRV
|
9.1 | IC50 | 8 | — | |
MTAOOMYAOJQXKB
|
9.1 | IC50 | 4 | — | |
BPBDCOLBZYWXHD
|
9.0 | IC50 | 24 | — | |
FMMIDZWTNQYEIY
|
9.0 | IC50 | 24 | — | |
JAWKANDWMZNIHM
|
9.0 | IC50 | 4 | — | |
JBHLOPKIPKTRSU
|
9.0 | Ki | 4 | — | |
RZEFTNLVGHECCN
|
9.0 | IC50 | 2 | — | |
VHBHGRJDLFMVBX
|
9.0 | IC50 | 2 | — | |
AZEXWHKOMMASPA
|
8.9 | IC50 | 2 | — | |
BWVJYTGTOWKCOX
|
8.8 | IC50 | 8 | — | |
NNRBBYSQRDRSCZ
|
8.8 | IC50 | 2 | — |