Target Details
| UniProt AC | Q9Y210 |
|---|---|
| Gene Symbol | TRPC6 |
| Protein Name | Short transient receptor potential channel 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12796 (Ank_2) PF00520 (Ion_trans) PF08344 (TRP_2) |
Summary
- Multi-target molecules 48
- Clinical molecules 0
- Avg pChEMBL 7.7
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (48)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MZAOLBDFKVMZHQ
|
8.6 | IC50 | 2 | — | |
KFJNTKXUHMJOFT
|
8.5 | IC50 | 2 | — | |
YYBCNHLZAHJUAY
|
8.5 | IC50 | 2 | — | |
WEKMAAKYOYJWIW
|
8.5 | IC50 | 2 | — | |
MWGNYVNFYUFWJE
|
8.4 | IC50 | 2 | — | |
GGKQWFQQUMWVOB
|
8.4 | IC50 | 2 | — | |
JIQJJGRQXFKITC
|
8.4 | IC50 | 2 | — | |
GAEQCZQSVPUDDV
|
8.3 | IC50 | 2 | — | |
VDWLBNKHHJKPOQ
|
8.2 | IC50 | 2 | — | |
NXPWFBZGNLXYOL
|
8.2 | IC50 | 2 | — | |
VNCKUJRDBRPUED
|
8.2 | IC50 | 2 | — | |
KKHVKJCJLDSGBE
|
8.1 | IC50 | 2 | — | |
ADSMSIAHGRRRDF
|
8.0 | IC50 | 2 | — | |
ODVBKRLGINBASD
|
8.0 | IC50 | 2 | — | |
RLKRLNQEXBPQGQ
|
8.0 | IC50 | 3 | — | |
UBMOUBBRNPNZPM
|
8.0 | IC50 | 2 | — | |
ZQPYFSHNTYXOFX
|
8.0 | IC50 | 2 | — | |
JTMAGZLVVBRGSP
|
8.0 | IC50 | 2 | — | |
YVAGLWQBGILNIU
|
8.0 | IC50 | 2 | — | |
KDEHDDNJCYLYNQ
|
7.9 | IC50 | 2 | — | |
PVEWBPFBLWIIRG
|
7.9 | IC50 | 2 | — | |
YSVYTXABMSDVMP
|
7.8 | IC50 | 2 | — | |
ODUIXUGXPFKQLG
|
7.8 | IC50 | 2 | — | |
OIKKWZUQICZOOT
|
7.8 | IC50 | 2 | — | |
LDMYUGCQIZOUKS
|
7.8 | IC50 | 2 | — | |
ATMDJXVKAVYNRI
|
7.8 | IC50 | 2 | — | |
WJUOPLMYEVNUCV
|
7.8 | IC50 | 2 | — | |
IKQBZXOTMPFTSS
|
7.8 | IC50 | 2 | — | |
ACTFBLSRASDXMR
|
7.7 | IC50 | 2 | — | |
CLBDHUXETCTAAC
|
7.7 | IC50 | 2 | — | |
ADSMSIAHGRRRDF
|
7.7 | IC50 | 2 | — | |
FWLXWTCADCXNQU
|
7.6 | IC50 | 2 | — | |
SEMFMCZEFJOTEB
|
7.6 | IC50 | 2 | — | |
KWHAFIYYZOUXKW
|
7.6 | IC50 | 2 | — | |
YWCKBHDCKIOOJA
|
7.5 | IC50 | 2 | — | |
ATVWXELBUSAQIM
|
7.5 | IC50 | 2 | — | |
KUVNZIJPYDWNHA
|
7.5 | IC50 | 2 | — | |
DXYANPCOKLRSRL
|
7.5 | IC50 | 2 | — | |
ODUIXUGXPFKQLG
|
7.3 | IC50 | 2 | — | |
ODUIXUGXPFKQLG
|
7.3 | IC50 | 2 | — | |
AOMYTFOGWHSXRM
|
7.2 | IC50 | 2 | — | |
YKFSMOUFOXUQLG
|
7.1 | IC50 | 2 | — | |
JFIIPBIYIJFPEE
|
6.8 | IC50 | 2 | — | |
VQYLWKAFQNHLFX
|
6.8 | IC50 | 2 | — | |
WORQHMTVOPUIRG
|
6.4 | IC50 | 2 | — | |
BQCVGSNZEUQCIS
|
6.2 | IC50 | 2 | — | |
QHHMGNMLPPWWIO
|
6.1 | IC50 | 2 | — | |
VEIFRHMKIXVPLN
|
6.1 | IC50 | 2 | — |