Target Details
| UniProt AC | Q9WKE8 |
|---|---|
| Gene Symbol | reverse transcriptase |
| Protein Name | N/A |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00078 (RVT_1) |
Summary
- Multi-target molecules 994
- Clinical molecules 0
- Avg pChEMBL 7.18
Active Molecules (994)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MZVNNERAAYHFPD
|
9.7 | IC50 | 2 | — | |
SVMHTBVIPYVDIL
|
9.6 | IC50 | 2 | — | |
KXDIHAQCVNNLIB
|
9.5 | IC50 | 2 | — | |
FKUXHXTYZGJMGB
|
9.4 | IC50 | 2 | — | |
RMXYGIHJODGJHN
|
9.4 | IC50 | 2 | — | |
JWDAEHXXNUMMKQ
|
9.4 | Ki | 2 | — | |
AASLKIYYTISYOA
|
9.3 | Ki | 2 | — | |
RURQSSZVFHRLEE
|
9.3 | Ki | 2 | — | |
PRHGIYDCDMLXHN
|
9.3 | IC50 | 2 | — | |
OCABMICVVJLNTB
|
9.2 | Ki | 2 | — | |
PCUWRGFJGCYISU
|
9.0 | IC50 | 2 | — | |
ATXSRWHPTOHHAY
|
9.0 | IC50 | 2 | — | |
FLGARVIJXJZDND
|
9.0 | IC50 | 2 | — | |
GUSPHNVTAWXCCQ
|
9.0 | IC50 | 2 | — | |
UOZDWSRONYZLQO
|
9.0 | IC50 | 2 | — | |
USWKTQVAABDFSY
|
9.0 | IC50 | 2 | — | |
BFPBNKBYNOBOHM
|
9.0 | IC50 | 2 | — | |
GCZMATZWHYCJTH
|
9.0 | IC50 | 2 | — | |
NKPHEWJJTGPRSL
|
9.0 | Kd | 2 | — | |
NPXCVIODFSNHMU
|
9.0 | IC50 | 2 | — | |
POOBUACLMWERDQ
|
9.0 | IC50 | 2 | — | |
UUVBMMWJHPNLHN
|
9.0 | IC50 | 2 | — | |
DTCDDPOBJLMFDD
|
8.9 | IC50 | 2 | — | |
PNJKKJNQGSBNDN
|
8.8 | IC50 | 2 | — | |
RTMMFLXVQPUVNI
|
8.8 | Ki | 2 | — | |
SSFUYPBGOTXADP
|
8.8 | IC50 | 2 | — | |
PMVRLVXVFQPYOQ
|
8.8 | Ki | 2 | — | |
DNNXGKQZFKHVRU
|
8.7 | IC50 | 2 | — | |
IDNIWMWKAMOXLP
|
8.7 | IC50 | 2 | — | |
NZABYUMWKMPSBX
|
8.7 | IC50 | 2 | — | |
SZLMFNKKFJUHKQ
|
8.7 | IC50 | 2 | — | |
YGWYLCTVXDISQZ
|
8.7 | IC50 | 2 | — | |
ZRYHQJAOERFYMX
|
8.7 | IC50 | 2 | — | |
JDPBFYPOTBVWBU
|
8.7 | Ki | 2 | — | |
QPIYUHRAHJHMRR
|
8.7 | Ki | 2 | — | |
SSUZBIFUDPSYGO
|
8.7 | IC50 | 2 | — | |
RGRSOJUFXZMIHM
|
8.7 | IC50 | 2 | — | |
GYBNBRVJAPRVLI
|
8.6 | IC50 | 2 | — | |
JFIAVEATUHYZRN
|
8.6 | IC50 | 2 | — | |
LPQYTOYTUGNTHQ
|
8.6 | IC50 | 2 | — | |
AVNBRYDGABAMIV
|
8.6 | Ki | 2 | — | |
KKDFGWKNYMTGFQ
|
8.6 | IC50 | 2 | — | |
USRHSVZSPKDGMT
|
8.6 | IC50 | 2 | — | |
GCSGUSKCFDTWJA
|
8.6 | IC50 | 2 | — | |
HKMAYQXCIOLGBJ
|
8.5 | IC50 | 2 | — | |
OKDKQGCRSIBHSQ
|
8.5 | IC50 | 2 | — | |
SXELKXZIKMONBL
|
8.5 | Ki | 2 | — | |
ANVDAXBIMHWBRJ
|
8.5 | IC50 | 2 | — | |
AWAKIULNKVOBKE
|
8.5 | IC50 | 2 | — | |
BEQOWVUOJYDODX
|
8.5 | IC50 | 2 | — |