Target Details
| UniProt AC | Q9WJQ2 |
|---|---|
| Gene Symbol | reverse transcriptase |
| Protein Name | N/A |
| Organism | Human immunodeficiency virus type 1 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00078 (RVT_1) |
Summary
- Multi-target molecules 144
- Clinical molecules 0
- Avg pChEMBL 7.66
Active Molecules (144)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AOIKBWIBFXPPRC
|
9.5 | IC50 | 2 | — | |
QWNIWQCTNAQHAF
|
9.4 | Ki | 2 | — | |
UMHXETHRMTWBPR
|
9.3 | Ki | 2 | — | |
FZBAOOQVQXATRL
|
9.2 | Ki | 2 | — | |
RXQSMZOUOHXYOX
|
9.1 | IC50 | 2 | — | |
YQELPLJAHMWKIX
|
9.0 | Ki | 2 | — | |
UMPSTPLBACSCDI
|
9.0 | IC50 | 2 | — | |
WHCLIFOVZDANCU
|
9.0 | IC50 | 2 | — | |
BUECGHMIFPUORL
|
8.9 | IC50 | 2 | — | |
SBDZLPIXOSPFIW
|
8.8 | IC50 | 2 | — | |
IJTWXTIWZPKVDV
|
8.8 | IC50 | 2 | — | |
ZSDYTNJSFLYICM
|
8.8 | Ki | 2 | — | |
ABOZXYNAPFTBHX
|
8.8 | Ki | 2 | — | |
RUEZUQUJOIHYNQ
|
8.8 | Ki | 2 | — | |
BTOMIMSUTLPSHA
|
8.8 | IC50 | 2 | — | |
KVJCKKKSJAZIHH
|
8.7 | IC50 | 2 | — | |
YCIPBZALVAZULV
|
8.7 | Ki | 2 | — | |
PJDCZSKXLVBCNA
|
8.6 | Ki | 2 | — | |
ZOPLPSKLHFWWGT
|
8.5 | IC50 | 2 | — | |
SQGNYTDBQSSZEE
|
8.5 | IC50 | 2 | — | |
BMOJLYKWVNBRLY
|
8.4 | IC50 | 2 | — | |
YMRUCOCNLHJFRC
|
8.4 | Ki | 2 | — | |
JPSHATBRSXMHDD
|
8.4 | Ki | 2 | — | |
IPURPIAIQWFSPQ
|
8.4 | IC50 | 2 | — | |
VMZCSGVUCCGELW
|
8.4 | IC50 | 2 | — | |
CUYHWBGVPXGMKQ
|
8.4 | Ki | 2 | — | |
QSAWJDNKFPMGBM
|
8.3 | Ki | 2 | — | |
ZFILMNZQPSHFSZ
|
8.3 | IC50 | 2 | — | |
QAPCSQPQKODCBU
|
8.3 | Ki | 2 | — | |
XIWJYQJWSFRHJL
|
8.3 | Ki | 2 | — | |
ALLQDFMKVJMXSZ
|
8.2 | IC50 | 2 | — | |
DCRLONDGVUVHIO
|
8.2 | IC50 | 2 | — | |
HHWIGJYKVRTBFJ
|
8.2 | IC50 | 2 | — | |
KLMNQDGJZUNXGC
|
8.2 | IC50 | 2 | — | |
AIFBSHYMNHBOFH
|
8.2 | IC50 | 2 | — | |
SBUMXUSAHHKUBE
|
8.2 | IC50 | 2 | — | |
MBIDFEZSWRDKLB
|
8.1 | IC50 | 2 | — | |
IHCSNCPUXYAQOH
|
8.1 | IC50 | 2 | — | |
URBRWOCTHYUBBB
|
8.1 | IC50 | 2 | — | |
JSTRBBFHRKOOAS
|
8.1 | IC50 | 2 | — | |
YZEAJCOIBSMIOB
|
8.1 | IC50 | 3 | — | |
JWSYHRYRAITBIX
|
8.0 | IC50 | 2 | — | |
UBXXFDJETHMQAG
|
8.0 | IC50 | 2 | — | |
GHQLRJSTAXRERC
|
7.9 | IC50 | 2 | — | |
NOIQCRFIOYMHLK
|
7.8 | IC50 | 2 | — | |
NPPGPCZJIKXPNW
|
7.8 | IC50 | 2 | — | |
GKFAGGGLMOZPIH
|
7.8 | IC50 | 2 | — | |
UFZKXRFAXDLHOV
|
7.8 | IC50 | 2 | — | |
USURLDWGSGIIKO
|
7.8 | IC50 | 2 | — | |
BAWWCXDEGWTQQJ
|
7.8 | IC50 | 2 | — |