Target Details
| UniProt AC | Q9UQM7 |
|---|---|
| Gene Symbol | CAMK2A |
| Protein Name | Calcium/calmodulin-dependent protein kinase type II subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08332 (CaMKII_AD) PF00069 (Pkinase) |
Summary
- Multi-target molecules 75
- Clinical molecules 31
- Avg pChEMBL 6.83
KEGG Pathways (34)
- Adrenergic signaling in cardiomyocytes
- Aldosterone synthesis and secretion
- Amphetamine addiction
- Axon guidance
- Calcium signaling pathway
- Cholinergic synapse
- Circadian entrainment
- Cushing syndrome
- Diabetic cardiomyopathy
- Dopaminergic synapse
- Efferocytosis
- ErbB signaling pathway
- Gastric acid secretion
- Glioma
- Glucagon signaling pathway
- GnRH signaling pathway
- HIF-1 signaling pathway
- Inflammatory mediator regulation of TRP channels
- Insulin secretion
- Lipid and atherosclerosis
- Long-term potentiation
- Melanogenesis
- Necroptosis
- Neurotrophin signaling pathway
- Olfactory transduction
- Oocyte meiosis
- Oxytocin signaling pathway
- Parkinson disease
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Proteoglycans in cancer
- Tuberculosis
- Wnt signaling pathway
- cAMP signaling pathway
Associated Diseases (2)
Active Molecules (75)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XUFLBSMTYMFOQH
|
6.4 | Ki | 43 | — | |
ZGZVRPRSFXRGCF
|
6.4 | Ki | 76 | — | |
NZXJTWVLQGCJJH
|
6.4 | IC50 | 7 | Yes | |
UIRCQOKSJDLYBB
|
6.3 | Ki | 50 | — | |
WAKGEHXTOOFEAE
|
6.3 | Ki | 27 | — | |
APPFRBZOALDJNI
|
6.3 | IC50 | 7 | Yes | |
SZJYMJNAWBOTEU
|
6.3 | IC50 | 9 | Yes | |
OWRXHGAFWZFFCW
|
6.2 | Ki | 113 | — | |
MRBBFOWSPXHYQT
|
6.2 | IC50 | 2 | — | |
ZZSBPGIGIUFJRA
|
6.2 | Kd | 46 | — | |
XCSNYNNJQSXDKR
|
6.1 | IC50 | 9 | Yes | |
SFDFKLDQKSPRHB
|
6.1 | IC50 | 15 | Yes | |
DFMCXVONDDGQIY
|
6.1 | Ki | 66 | — | |
MSEGDVOYFLNBPZ
|
6.1 | IC50 | 2 | — | |
ADQKGRUFGPUORP
|
6.0 | IC50 | 9 | Yes | |
QQWUGDVOUVUTOY
|
6.0 | Kd | 231 | Yes | |
GJOXRIYWDHESDF
|
6.0 | Ki | 27 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
OHNNRNYUHNGDNO
|
6.0 | IC50 | 15 | — | |
QVNZKVACBBTKSL
|
6.0 | Ki | 38 | — | |
RZJKNYACYSIBFY
|
6.0 | IC50 | 4 | — | |
SDTHQOXRWZXTJF
|
6.0 | Ki | 16 | — | |
XTVULKIROSNNTG
|
6.0 | Ki | 29 | — | |
YYPKOMNJRZRWIC
|
6.0 | Ki | 26 | — | |
ZHJGWYRLJUCMRT
|
6.0 | Kd | 18 | — |