Target Details
| UniProt AC | Q9UQM7 |
|---|---|
| Gene Symbol | CAMK2A |
| Protein Name | Calcium/calmodulin-dependent protein kinase type II subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08332 (CaMKII_AD) PF00069 (Pkinase) |
Summary
- Multi-target molecules 75
- Clinical molecules 31
- Avg pChEMBL 6.83
KEGG Pathways (34)
- Adrenergic signaling in cardiomyocytes
- Aldosterone synthesis and secretion
- Amphetamine addiction
- Axon guidance
- Calcium signaling pathway
- Cholinergic synapse
- Circadian entrainment
- Cushing syndrome
- Diabetic cardiomyopathy
- Dopaminergic synapse
- Efferocytosis
- ErbB signaling pathway
- Gastric acid secretion
- Glioma
- Glucagon signaling pathway
- GnRH signaling pathway
- HIF-1 signaling pathway
- Inflammatory mediator regulation of TRP channels
- Insulin secretion
- Lipid and atherosclerosis
- Long-term potentiation
- Melanogenesis
- Necroptosis
- Neurotrophin signaling pathway
- Olfactory transduction
- Oocyte meiosis
- Oxytocin signaling pathway
- Parkinson disease
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Proteoglycans in cancer
- Tuberculosis
- Wnt signaling pathway
- cAMP signaling pathway
Associated Diseases (2)
Active Molecules (75)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
9.9 | IC50 | 408 | — | |
HKSZLNNOFSGOKW
|
9.8 | Kd | 213 | — | |
HKSZLNNOFSGOKW
|
8.5 | Ki | 118 | — | |
GDQXJQSQYMMKRA
|
8.1 | IC50 | 15 | — | |
OSVUGUHRKMMBSE
|
8.1 | Kd | 170 | — | |
UIARLYUEJFELEN
|
8.0 | Kd | 289 | Yes | |
NXSJMRCTGYTSTK
|
7.8 | Kd | 200 | — | |
BMGQWWVMWDBQGC
|
7.7 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
7.7 | Kd | 91 | Yes | |
KAJXOWFGKYKMMZ
|
7.6 | IC50 | 26 | Yes | |
LEJHMQJABOLACY
|
7.6 | IC50 | 9 | Yes | |
KSILWADEZRASEE
|
7.5 | IC50 | 4 | — | |
NOVLXWHGKLXEJS
|
7.4 | IC50 | 4 | — | |
RGNHKJWHFIPHIM
|
7.4 | Ki | 66 | — | |
APALQVMWCDGRJB
|
7.3 | IC50 | 9 | Yes | |
HFNKQEVNSGCOJV
|
7.3 | Kd | 65 | — | |
ZNEQEOGXKINPPR
|
7.3 | IC50 | 9 | Yes | |
LAMWYYXJYIQOQL
|
7.2 | IC50 | 16 | Yes | |
GPNZOTCLQNMQIC
|
7.2 | IC50 | 7 | Yes | |
NWMPVMMGSHXANZ
|
7.2 | Ki | 58 | — | |
CMWRPDHVGMHLSZ
|
7.2 | IC50 | 22 | — | |
WINHZLLDWRZWRT
|
7.1 | Kd | 201 | Yes | |
XOFQJBDORDALAH
|
7.1 | IC50 | 9 | Yes | |
ZPEBZVFGLUUCDX
|
7.1 | IC50 | 6 | — | |
WMUGNCAVDUVWIE
|
7.0 | IC50 | 9 | Yes | |
CHOKPCNUYFDUDO
|
7.0 | IC50 | 9 | Yes | |
BRGYPSBHCUNPNP
|
7.0 | IC50 | 9 | Yes | |
XSHQBIXMLULFEV
|
7.0 | IC50 | 13 | — | |
AEYLJTAIDDIOBA
|
6.8 | Ki | 53 | — | |
FUMCKNCUEAQHCV
|
6.8 | Ki | 103 | — | |
WINHZLLDWRZWRT
|
6.8 | Ki | 66 | — | |
DJKBFCHOHWZUOH
|
6.8 | IC50 | 7 | Yes | |
SFQZZXBCKCLFFC
|
6.8 | IC50 | 6 | — | |
BDOCJJUGIOCUKN
|
6.8 | IC50 | 7 | Yes | |
MEXUTNIFSHFQRG
|
6.7 | IC50 | 21 | Yes | |
WDARYLSSWBWVCU
|
6.7 | Ki | 49 | — | |
ZGDYBJXDIXVTLV
|
6.7 | Ki | 54 | — | |
SDUWPCYMTHMQAZ
|
6.7 | IC50 | 8 | Yes | |
HFNKQEVNSGCOJV
|
6.7 | Ki | 18 | — | |
RPSCADUVKLRNEB
|
6.6 | IC50 | 8 | Yes | |
HZPACYSNLOCDLW
|
6.6 | Ki | 48 | — | |
ZHBAGBACXDDSPH
|
6.6 | IC50 | 9 | Yes | |
LKLASFRCXLTNMY
|
6.5 | IC50 | 4 | Yes | |
GGUSTVFLQLGLJX
|
6.5 | IC50 | 7 | Yes | |
JOOXLOJCABQBSG
|
6.5 | Kd | 139 | — | |
BPNUQXPIQBZCMR
|
6.5 | Kd | 83 | Yes | |
LBVKEEFIPBQIMD
|
6.5 | Ki | 27 | — | |
CTNPALGJUAXMMC
|
6.5 | Kd | 151 | — | |
ATHMTZOFUCSRPV
|
6.4 | IC50 | 7 | Yes | |
LHQWPYOYDRVMFI
|
6.4 | Ki | 21 | — |