Target Details
| UniProt AC | Q9UQD0 |
|---|---|
| Gene Symbol | SCN8A |
| Protein Name | Sodium channel protein type 8 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 272
- Clinical molecules 0
- Avg pChEMBL 7.06
KEGG Pathways (1)
Associated Diseases (4)
Active Molecules (272)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OHPHZNJGEVSWMX
|
6.2 | IC50 | 2 | — | |
HSOCYPPAQYZHMJ
|
6.2 | IC50 | 2 | — | |
JIEBHKJKDRMVCK
|
6.2 | IC50 | 2 | — | |
PKBLNJQHGWHMLE
|
6.2 | IC50 | 2 | — | |
PNSVJQJVGCLXPD
|
6.2 | IC50 | 2 | — | |
VUXLKOATKUTQHW
|
6.2 | IC50 | 3 | — | |
YDRSKXBOYKSOJN
|
6.2 | IC50 | 2 | — | |
LWWSUXPACZILER
|
6.1 | IC50 | 2 | — | |
QNKJHZQKTGVKRT
|
6.1 | IC50 | 2 | — | |
REFSPUPAKCCVAD
|
6.1 | IC50 | 2 | — | |
VVSUNZXJDARYBH
|
6.1 | IC50 | 2 | — | |
SZDIBDVGYBSTGV
|
6.1 | IC50 | 2 | — | |
AWWVNDFZXGVFPE
|
6.1 | IC50 | 2 | — | |
AYTPMWAPDMTVKH
|
6.1 | IC50 | 2 | — | |
SVHFOHFXYDMAPK
|
6.1 | IC50 | 2 | — | |
KZMGUTIQLABKCR
|
6.1 | IC50 | 2 | — | |
SUDPZTYFJSTPQI
|
6.0 | IC50 | 2 | — | |
MULKIBHRPCRKGZ
|
6.0 | IC50 | 2 | — | |
LVBOJKUDPCHPOK
|
6.0 | IC50 | 2 | — | |
HBNPJJILLOYFJU
|
6.0 | IC50 | 21 | — | |
QJETWCFGSMIKHY
|
6.0 | IC50 | 2 | — | |
WMZBZYXATSTGOK
|
6.0 | IC50 | 2 | — |