Target Details
| UniProt AC | Q9UQD0 |
|---|---|
| Gene Symbol | SCN8A |
| Protein Name | Sodium channel protein type 8 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 272
- Clinical molecules 0
- Avg pChEMBL 7.06
KEGG Pathways (1)
Associated Diseases (4)
Active Molecules (272)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZENFAJIAXHLNGU
|
6.6 | IC50 | 2 | — | |
VVLOWQFWNDSOLZ
|
6.6 | IC50 | 2 | — | |
VXMXACPWGGRFIF
|
6.5 | IC50 | 2 | — | |
XBCPDKDJZGECMM
|
6.5 | IC50 | 2 | — | |
QKQXMYZOQMBBRN
|
6.5 | IC50 | 2 | — | |
YEDAUVHICLPEIJ
|
6.5 | IC50 | 2 | — | |
LNRALXGEGPHUEQ
|
6.5 | IC50 | 2 | — | |
ODABGVBBVPDXSL
|
6.5 | IC50 | 2 | — | |
SRJPMKIXDZZWAT
|
6.5 | IC50 | 2 | — | |
UUJCWXBORMXXGI
|
6.5 | IC50 | 2 | — | |
URZHGUANLMQVBE
|
6.5 | IC50 | 2 | — | |
LGABDIUYXJPBQQ
|
6.5 | IC50 | 2 | — | |
BXOIJQLSRAKHJK
|
6.5 | IC50 | 2 | — | |
CGHVTPLFSBFCMC
|
6.5 | IC50 | 2 | — | |
CRIVLAVCQBIGSC
|
6.5 | IC50 | 2 | — | |
ZDKAXYKVNSBOHU
|
6.5 | IC50 | 2 | — | |
JYSHLENEZRKPDK
|
6.5 | IC50 | 2 | — | |
XUGUKAXHZIOGLG
|
6.5 | IC50 | 2 | — | |
OFVXFYHEMPXWQX
|
6.5 | IC50 | 2 | — | |
PXKQOZLVZUDGPQ
|
6.5 | IC50 | 2 | — | |
QYTIKFWKCOVLGN
|
6.5 | IC50 | 2 | — | |
SHUSNHMECJFRFW
|
6.4 | IC50 | 2 | — | |
FJCCQQXMASEMDV
|
6.4 | IC50 | 2 | — | |
QJYSAPCKCOXUFR
|
6.4 | IC50 | 2 | — | |
QCDCHYCAWONKAY
|
6.4 | IC50 | 2 | — | |
HPURRFIKNKVIFS
|
6.4 | IC50 | 2 | — | |
KLWKJFRXLGLTIH
|
6.4 | IC50 | 4 | — | |
ONNZXUHXIVNZBQ
|
6.4 | IC50 | 2 | — | |
GVGBKXMUVOMTDB
|
6.4 | IC50 | 2 | — | |
PKVSOUFAHPBDDR
|
6.4 | IC50 | 2 | — | |
MWDAENLOSFCPCZ
|
6.4 | IC50 | 2 | — | |
IDVVCBYQIPGRMK
|
6.3 | IC50 | 2 | — | |
QUPOUNZWMBLXGJ
|
6.3 | IC50 | 2 | — | |
RVSQXLHJPFTVRX
|
6.3 | IC50 | 2 | — | |
CZGJOHTUWRUTMS
|
6.3 | IC50 | 2 | — | |
FBTZFSFVDPEXDW
|
6.3 | IC50 | 2 | — | |
OTBNOCRUGHNICR
|
6.3 | IC50 | 2 | — | |
VJQQATGQOSVQCZ
|
6.3 | IC50 | 2 | — | |
IQNGIYJIIGTIOM
|
6.3 | IC50 | 2 | — | |
JYEYDNUQQSHVRP
|
6.3 | IC50 | 2 | — | |
OJKONCJPCULNOW
|
6.3 | IC50 | 4 | — | |
PTCBNPULJWGSML
|
6.3 | IC50 | 9 | — | |
FCWGDENQRAUXMY
|
6.3 | IC50 | 2 | — | |
KICOFBPOACPQPG
|
6.3 | IC50 | 2 | — | |
BVJWKHFIJISOQD
|
6.3 | IC50 | 2 | — | |
KUEGRSXKAHKHIA
|
6.3 | IC50 | 5 | — | |
GKCBAIGFKIBETG
|
6.3 | IC50 | 10 | — | |
DITZNZYXKSFLJE
|
6.2 | IC50 | 2 | — | |
BSCTXVDJXNZALB
|
6.2 | IC50 | 2 | — | |
KQQXPTRMUYKUIC
|
6.2 | Kd | 8 | — |