Target Details
| UniProt AC | Q9UQD0 |
|---|---|
| Gene Symbol | SCN8A |
| Protein Name | Sodium channel protein type 8 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 272
- Clinical molecules 0
- Avg pChEMBL 7.06
KEGG Pathways (1)
Associated Diseases (4)
Active Molecules (272)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UTKZKXRKSFATLD
|
7.0 | IC50 | 2 | — | |
ALYSSPGOUMAGSF
|
7.0 | IC50 | 5 | — | |
YURAPCXMUFFHQV
|
7.0 | IC50 | 2 | — | |
CEWKJGUDXOKCAF
|
7.0 | IC50 | 2 | — | |
MFOFLSYIDKCECT
|
7.0 | IC50 | 2 | — | |
BKBBARITZRESJB
|
6.9 | IC50 | 2 | — | |
HGWQEYGUKORMFX
|
6.9 | IC50 | 2 | — | |
UEAQPOVLANIUKN
|
6.9 | IC50 | 2 | — | |
ZBHRJPDUINZSBQ
|
6.9 | IC50 | 2 | — | |
GJSPKAUMUKBENE
|
6.9 | IC50 | 2 | — | |
ICYNQJUIRKNXOK
|
6.9 | IC50 | 2 | — | |
KYRYYQRTAJIXDA
|
6.9 | IC50 | 2 | — | |
NCFGRWURVNNKRV
|
6.9 | IC50 | 2 | — | |
NJMQDDCKQPGJLM
|
6.9 | IC50 | 2 | — | |
ZXKIOHRLQVWVGA
|
6.9 | IC50 | 2 | — | |
DFBDAHMZXJYZJG
|
6.9 | IC50 | 7 | — | |
OHPHZNJGEVSWMX
|
6.9 | IC50 | 2 | — | |
WTPNXRKKYIAOOU
|
6.9 | IC50 | 2 | — | |
IXFWXFPSQUGQID
|
6.9 | IC50 | 2 | — | |
KUCYRCUGXDBLAO
|
6.9 | IC50 | 2 | — | |
QFNICIAXNSXIJO
|
6.8 | IC50 | 2 | — | |
JIKVCZBAPMSLIV
|
6.8 | IC50 | 2 | — | |
UJNYFUQRHSEWMI
|
6.8 | IC50 | 2 | — | |
IKWWVCWYCSDROX
|
6.8 | IC50 | 2 | — | |
JWBFMRPLLUIRBB
|
6.8 | IC50 | 2 | — | |
KJFXVAHPAFFCTE
|
6.8 | IC50 | 2 | — | |
BDNWHXABGMGJIY
|
6.8 | IC50 | 2 | — | |
MJJULZATLMLYAP
|
6.8 | IC50 | 2 | — | |
NRKTYVBSUNDFEM
|
6.8 | IC50 | 2 | — | |
ZYSCOUXLBXGGIM
|
6.8 | IC50 | 9 | — | |
NEBUOXBYNAHKFV
|
6.8 | IC50 | 5 | — | |
AAUMZZJEGXJINE
|
6.7 | IC50 | 3 | — | |
PNKCJCUVBPXLEN
|
6.7 | IC50 | 2 | — | |
DPGOQYYAHWEROP
|
6.7 | IC50 | 5 | — | |
FVGGAZKZIUTNLQ
|
6.7 | IC50 | 5 | — | |
SXOAHIZWCZOILH
|
6.7 | IC50 | 9 | — | |
IJZKTKBPFIPSJP
|
6.7 | IC50 | 2 | — | |
KYBPOTYVFWNSGS
|
6.7 | Kd | 8 | — | |
OEQKFOZNCUDRFU
|
6.7 | IC50 | 2 | — | |
YYEFHRUFIOSDKV
|
6.7 | IC50 | 2 | — | |
PUIQVUPDIYCXBY
|
6.7 | IC50 | 2 | — | |
XNDLSZOBHUFYDN
|
6.7 | IC50 | 2 | — | |
NNOURUCQGKSLJV
|
6.6 | IC50 | 2 | — | |
RGBIVRJIERNIRK
|
6.6 | IC50 | 2 | — | |
RXHXBPPRDMVRJS
|
6.6 | IC50 | 2 | — | |
QUJPVMQGTDABGN
|
6.6 | IC50 | 2 | — | |
AOAGKSSQGPUXSO
|
6.6 | IC50 | 2 | — | |
XEDSOXUCOFSPMG
|
6.6 | IC50 | 2 | — | |
KPACYEJRAQEPQE
|
6.6 | IC50 | 2 | — | |
TTXHVPIJWCJKLK
|
6.6 | IC50 | 2 | — |