Target Details
| UniProt AC | Q9UQD0 |
|---|---|
| Gene Symbol | SCN8A |
| Protein Name | Sodium channel protein type 8 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 272
- Clinical molecules 0
- Avg pChEMBL 7.06
KEGG Pathways (1)
Associated Diseases (4)
Active Molecules (272)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TXAYOTYZKGQCMM
|
7.2 | IC50 | 2 | — | |
ZBIVKTYZIJLJTE
|
7.2 | IC50 | 2 | — | |
GFSUVQOECDPIQJ
|
7.2 | IC50 | 4 | — | |
GOXQSPDBNHQSLA
|
7.2 | IC50 | 2 | — | |
IHXQTRXZYHPGIQ
|
7.2 | IC50 | 2 | — | |
KTUKIQYULOKPOV
|
7.2 | IC50 | 4 | — | |
XMZFDPKNGIFRLZ
|
7.2 | IC50 | 2 | — | |
DVXZPBHBSUZGDY
|
7.2 | IC50 | 2 | — | |
VEEQSZWXUOUXPZ
|
7.2 | IC50 | 5 | — | |
GFDFBVYVIAOKEU
|
7.2 | IC50 | 2 | — | |
CUVWAXHFLWGMGR
|
7.2 | IC50 | 2 | — | |
ICZIAJCVIIUREC
|
7.2 | IC50 | 2 | — | |
QDWZJQPXKINAHW
|
7.2 | IC50 | 2 | — | |
XQOGUSYHWGLZNJ
|
7.2 | IC50 | 2 | — | |
CQLAPNTWQQWKFV
|
7.2 | IC50 | 2 | — | |
IRHNPUOYGLVXGO
|
7.1 | IC50 | 2 | — | |
OSVWTSSVVMEISV
|
7.1 | IC50 | 2 | — | |
AWXDDGVMVDUNGA
|
7.1 | IC50 | 2 | — | |
PSTCCBODERRWFK
|
7.1 | IC50 | 2 | — | |
NDMNISGHBWDHTB
|
7.1 | IC50 | 2 | — | |
VRUSWBLOISBSSJ
|
7.1 | IC50 | 5 | — | |
CKTPSKKTZVSXLI
|
7.1 | IC50 | 2 | — | |
ACYYAPDBAJQILC
|
7.1 | IC50 | 2 | — | |
KEFLKWVDEZWQCI
|
7.1 | IC50 | 2 | — | |
QTEMPVGNCZGUQZ
|
7.1 | IC50 | 2 | — | |
HBBSMJFEJAGCAU
|
7.1 | IC50 | 2 | — | |
FWASJBQVSBHBNK
|
7.1 | IC50 | 2 | — | |
KPWHRDZTQCXAAK
|
7.0 | IC50 | 2 | — | |
ANGUVPSJNSWBFO
|
7.0 | IC50 | 4 | — | |
AQMSMCUTJNXRFL
|
7.0 | IC50 | 2 | — | |
FPERPEQIXLOVIK
|
7.0 | IC50 | 5 | — | |
HCOYRSDKPDEDHP
|
7.0 | IC50 | 2 | — | |
NNYFWIVNWYRZQL
|
7.0 | IC50 | 2 | — | |
GHXUGFVKIDRBGU
|
7.0 | IC50 | 2 | — | |
PDRLXIQAZYHBJG
|
7.0 | IC50 | 2 | — | |
QLJAUMYWJMHEIG
|
7.0 | IC50 | 2 | — | |
ROWKGBJMLVUFFH
|
7.0 | IC50 | 2 | — | |
YMFGIDHGVTYYJZ
|
7.0 | IC50 | 2 | — | |
UMDJUPAXVBHNKS
|
7.0 | IC50 | 2 | — | |
FQRONRPRMDEQNS
|
7.0 | IC50 | 2 | — | |
IBHSESFTJVMJEA
|
7.0 | IC50 | 2 | — | |
MASHRDPYQKFCAR
|
7.0 | IC50 | 2 | — | |
OHPHZNJGEVSWMX
|
7.0 | IC50 | 2 | — | |
ZKNUWIKFMSHCTJ
|
7.0 | IC50 | 2 | — | |
ZXMZQSSITMSTKQ
|
7.0 | IC50 | 2 | — | |
JCPHCHCAKXVPLC
|
7.0 | IC50 | 2 | — | |
SUDPJHWRLKPICV
|
7.0 | IC50 | 3 | — | |
CBWXHMITTMOYOY
|
7.0 | IC50 | 2 | — | |
OVWZROCNURWRKK
|
7.0 | IC50 | 2 | — | |
PRDWHZNGVONJAX
|
7.0 | IC50 | 2 | — |