Target Details
| UniProt AC | Q9UQD0 |
|---|---|
| Gene Symbol | SCN8A |
| Protein Name | Sodium channel protein type 8 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 272
- Clinical molecules 0
- Avg pChEMBL 7.06
KEGG Pathways (1)
Associated Diseases (4)
Active Molecules (272)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XQUOWYVEKSXNET
|
7.5 | Kd | 3 | — | |
YNWHWKIVLFOBNC
|
7.5 | IC50 | 2 | — | |
FZRXMWNNMIDCAX
|
7.5 | IC50 | 2 | — | |
HBBSMJFEJAGCAU
|
7.5 | IC50 | 2 | — | |
POWGSPMXXFULOC
|
7.5 | IC50 | 2 | — | |
XFYJZSKHXSPHJR
|
7.5 | IC50 | 2 | — | |
IVXWSJDIJWTMBP
|
7.5 | IC50 | 2 | — | |
OFZBNADUYSHVNR
|
7.5 | IC50 | 2 | — | |
YVVIILBXFPZWHI
|
7.5 | IC50 | 2 | — | |
YFLRARPBRFARON
|
7.5 | IC50 | 2 | — | |
ZKBINYGXHLBBGG
|
7.5 | IC50 | 2 | — | |
FECNWUDMIMNVGT
|
7.5 | IC50 | 2 | — | |
UEAAJOBUYFZGHL
|
7.5 | IC50 | 2 | — | |
KWARURQEBURTJY
|
7.5 | IC50 | 2 | — | |
YWQDQDUGUYEIPV
|
7.4 | IC50 | 2 | — | |
LPALDPYBGGHZSG
|
7.4 | IC50 | 2 | — | |
YSGJURKDIMZYFR
|
7.4 | IC50 | 2 | — | |
ZRKHPQPMAITAEP
|
7.4 | IC50 | 2 | — | |
GFDXIUXAFNREKM
|
7.4 | IC50 | 6 | — | |
DMQWJYJEJRIDBI
|
7.4 | IC50 | 2 | — | |
PGAFBTBFTNJDLQ
|
7.4 | IC50 | 3 | — | |
UXNUHKSSUVUOKZ
|
7.4 | IC50 | 2 | — | |
VOJFVKGTRNXOTJ
|
7.4 | IC50 | 4 | — | |
PKHVECBKGBDQAY
|
7.4 | IC50 | 2 | — | |
SXHSUVHECGYYMY
|
7.4 | IC50 | 2 | — | |
NVPMWUPUWBXETR
|
7.4 | IC50 | 2 | — | |
FPKSPIQOEJACSE
|
7.4 | IC50 | 2 | — | |
HAHBYABDAIXZLF
|
7.4 | IC50 | 2 | — | |
PIQAUSNVLROXMR
|
7.4 | IC50 | 2 | — | |
GGKJOYYMGVWXAT
|
7.3 | IC50 | 2 | — | |
IWRIRVFYRTUDIJ
|
7.3 | IC50 | 2 | — | |
BMYFAIFEOQGCTL
|
7.3 | IC50 | 2 | — | |
RFLSHFCTAZELPZ
|
7.3 | IC50 | 2 | — | |
XUCXIMYTIQZZHZ
|
7.3 | IC50 | 5 | — | |
JLOCNBNTRGBNSU
|
7.3 | IC50 | 2 | — | |
SDPRTZGVTOHKRX
|
7.3 | IC50 | 2 | — | |
IJLRJKVKJNUIJD
|
7.3 | IC50 | 2 | — | |
NUHUWFKTWWXUTJ
|
7.3 | IC50 | 2 | — | |
VWKUYSDQOUJGJG
|
7.3 | IC50 | 2 | — | |
YNXDPYBMQUPNTL
|
7.3 | IC50 | 2 | — | |
AXDMEYZFXMOJQC
|
7.3 | IC50 | 2 | — | |
AKDINRARGVIZNO
|
7.3 | IC50 | 2 | — | |
URUKPZGNTWPRGW
|
7.3 | IC50 | 2 | — | |
WGGALQWPTKGQLX
|
7.3 | IC50 | 2 | — | |
YVUQSNJEYSNKRX
|
7.3 | IC50 | 36 | — | |
IMKFJSDSDZBSQO
|
7.3 | IC50 | 2 | — | |
FAHBRZBMNSAQQB
|
7.2 | IC50 | 2 | — | |
HAHBFCDZJMZPDT
|
7.2 | IC50 | 2 | — | |
UFVVLUUDTNDRGT
|
7.2 | IC50 | 2 | — | |
MUUIZCFCJVLOGF
|
7.2 | IC50 | 2 | — |