Target Details
| UniProt AC | Q9UQD0 |
|---|---|
| Gene Symbol | SCN8A |
| Protein Name | Sodium channel protein type 8 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) PF11933 (Na_trans_cytopl) |
Summary
- Multi-target molecules 272
- Clinical molecules 0
- Avg pChEMBL 7.06
KEGG Pathways (1)
Associated Diseases (4)
Active Molecules (272)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XFWKBJBSEOZBRA
|
10.2 | IC50 | 3 | — | |
XBIMZDZZPNFVOV
|
10.1 | IC50 | 2 | — | |
NLTQZTZBFNPMDH
|
9.1 | IC50 | 3 | — | |
CSKLRKQUNQCFCW
|
9.0 | IC50 | 2 | — | |
GYAAKIKKAKLXDK
|
9.0 | IC50 | 2 | — | |
RPQXVSUAYFXFJA
|
9.0 | IC50 | 8 | — | |
TXMZTVOEZCLPIF
|
8.8 | IC50 | 2 | — | |
OZJSEVZVZWZBIT
|
8.7 | IC50 | 2 | — | |
CFMYXEVWODSLAX
|
8.6 | IC50 | 8 | — | |
XNAAGHKLQDFJAV
|
8.5 | IC50 | 2 | — | |
XBIMZDZZPNFVOV
|
8.3 | IC50 | 2 | — | |
OFJWZNKJBMVLPX
|
8.3 | IC50 | 2 | — | |
WSPHMGORSRQULF
|
8.2 | IC50 | 6 | — | |
MEEMNCAUXAWBBT
|
8.2 | IC50 | 2 | — | |
DSGSRMJPDQBTMM
|
8.2 | IC50 | 2 | — | |
ZPEBBZMLDYXDOW
|
8.0 | IC50 | 2 | — | |
OJGBGGHWKBSYTM
|
8.0 | IC50 | 2 | — | |
CYBITNCPJFQMIJ
|
8.0 | IC50 | 5 | — | |
INIMUMMAVCNJFA
|
8.0 | IC50 | 2 | — | |
JKAMBBDGLZFTHQ
|
8.0 | IC50 | 2 | — | |
QYLLDXJQSXDYLQ
|
8.0 | IC50 | 2 | — | |
AJZDQSWVXBSGJM
|
7.9 | IC50 | 2 | — | |
IDCLDFZOZFUTLI
|
7.9 | IC50 | 2 | — | |
UHWLWOOUNBNZHS
|
7.9 | IC50 | 2 | — | |
KZBXVOINEPFFDK
|
7.9 | IC50 | 2 | — | |
UUAIQHMLXPMLDV
|
7.8 | IC50 | 2 | — | |
YXHMFJXQQXHKRO
|
7.8 | IC50 | 2 | — | |
OGNHUCWKIBGDPU
|
7.8 | IC50 | 2 | — | |
ZUFQSMFAKHTNSW
|
7.8 | IC50 | 2 | — | |
PHXPCSYUXAKISO
|
7.8 | IC50 | 2 | — | |
GOHNZFHVWZRGGX
|
7.7 | IC50 | 2 | — | |
JXYDAQZEKBXJFK
|
7.7 | IC50 | 2 | — | |
WLRVZQGFKCYIOQ
|
7.7 | IC50 | 2 | — | |
WSAJJTWYTKFRMU
|
7.7 | IC50 | 2 | — | |
OJJVDLJKYRQHKJ
|
7.7 | IC50 | 2 | — | |
JEQHYRZPVUELSI
|
7.6 | IC50 | 2 | — | |
JNNYSEIQBAVVNL
|
7.6 | IC50 | 2 | — | |
KBLIOLOEZADQDG
|
7.6 | IC50 | 3 | — | |
LNYJTKCHVILHMC
|
7.6 | IC50 | 2 | — | |
LTPHTGJIOPSZAL
|
7.6 | IC50 | 2 | — | |
MLUQPNYVJYPKKO
|
7.6 | IC50 | 2 | — | |
GFUFBVLEJPJQBR
|
7.6 | IC50 | 2 | — | |
GIJKDQHCVRCMIN
|
7.6 | IC50 | 2 | — | |
IYMXTVBKMMBTML
|
7.6 | IC50 | 2 | — | |
LXEYTAIEXPOZNY
|
7.6 | IC50 | 2 | — | |
XLENMSSHHOXWHN
|
7.6 | IC50 | 2 | — | |
BVWMEUDWRCWKGL
|
7.5 | IC50 | 2 | — | |
FBEKVCAOQKXVOK
|
7.5 | IC50 | 2 | — | |
XENPFDQDTNUZPA
|
7.5 | IC50 | 2 | — | |
XOAUGYVLRSCGBG
|
7.5 | IC50 | 8 | — |