Target Details
| UniProt AC | Q9UQB9 |
|---|---|
| Gene Symbol | AURKC |
| Protein Name | Aurora kinase C |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 80
- Clinical molecules 25
- Avg pChEMBL 7.38
Associated Diseases (1)
Active Molecules (80)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OBWNXGOQPLDDPS
|
6.9 | IC50 | 6 | Yes | |
NVLLVQNRIGNKPZ
|
6.9 | IC50 | 3 | — | |
SHPFDGWALWEPGS
|
6.8 | Kd | 35 | — | |
LFKPJUFFMOTFRX
|
6.8 | IC50 | 6 | — | |
BMGQWWVMWDBQGC
|
6.8 | Kd | 147 | Yes | |
XZXHXSATPCNXJR
|
6.7 | Kd | 165 | Yes | |
MLDQJTXFUGDVEO
|
6.7 | Kd | 85 | Yes | |
NHFDRBXTEDBWCZ
|
6.7 | IC50 | 12 | Yes | |
WINHZLLDWRZWRT
|
6.7 | Kd | 201 | Yes | |
RXPZOSHFGJWSLQ
|
6.6 | IC50 | 6 | — | |
MRITYVDXXFOOAU
|
6.5 | Kd | 6 | — | |
QKKIWEILHCXECO
|
6.5 | IC50 | 24 | — | |
FQCPPVRJPILDIK
|
6.5 | IC50 | 12 | — | |
OYONTEXKYJZFHA
|
6.5 | Kd | 69 | Yes | |
DDLZLOKCJHBUHD
|
6.5 | IC50 | 23 | — | |
JOOXLOJCABQBSG
|
6.5 | Kd | 139 | — | |
PXGLIUGVLBRUBV
|
6.4 | IC50 | 3 | — | |
AKSIZPIFQAYJGF
|
6.4 | IC50 | 4 | Yes | |
HHJSKDRCUMVWKF
|
6.3 | IC50 | 7 | — | |
RKBMAROJKLHAMI
|
6.3 | IC50 | 6 | — | |
HDAJDNHIBCDLQF
|
6.2 | IC50 | 14 | — | |
ZHOXAGNPCZTRBN
|
6.2 | Kd | 20 | — | |
KTUZOTUSWXJDIS
|
6.2 | IC50 | 3 | — | |
AAKJLRGGTJKAMG
|
6.2 | Kd | 50 | Yes | |
ODPGGGTTYSGTGO
|
6.1 | Kd | 153 | — | |
CUIHSIWYWATEQL
|
6.1 | Kd | 61 | Yes | |
ZZSBPGIGIUFJRA
|
6.1 | Kd | 46 | — | |
CTNPALGJUAXMMC
|
6.1 | Kd | 151 | — | |
CURXWONZHCZVOV
|
6.0 | IC50 | 5 | — | |
NSMOZFXKTHCPTQ
|
6.0 | IC50 | 4 | — |