Target Details
| UniProt AC | Q9UQB9 |
|---|---|
| Gene Symbol | AURKC |
| Protein Name | Aurora kinase C |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 80
- Clinical molecules 25
- Avg pChEMBL 7.38
Associated Diseases (1)
Active Molecules (80)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BRXHKUKMMZTVRE
|
9.0 | IC50 | 3 | — | |
HOCURELMRBRHRJ
|
9.0 | Kd | 3 | — | |
IVUGFMLRJOCGAS
|
9.0 | IC50 | 9 | — | |
RITAVMQDGBJQJZ
|
8.9 | Kd | 43 | — | |
FZVCMCRNWSWUCG
|
8.7 | Kd | 3 | — | |
KZBSEJKXWKPCLO
|
8.7 | Kd | 3 | — | |
DQRVOAFQMMLWCP
|
8.5 | Kd | 3 | — | |
FAYAUAZLLLJJGH
|
8.5 | IC50 | 36 | Yes | |
XQNMCONHYXAHKS
|
8.5 | IC50 | 3 | — | |
QTBWCSQGBMPECM
|
8.5 | IC50 | 21 | Yes | |
NOHJLJNUPONZRF
|
8.4 | Kd | 3 | — | |
UIARLYUEJFELEN
|
8.4 | Kd | 289 | Yes | |
QYZOGCMHVIGURT
|
8.4 | Kd | 26 | Yes | |
GCIKSSRWRFVXBI
|
8.3 | Ki | 109 | Yes | |
WNQHVGYFQUHRNW
|
8.3 | Ki | 4 | — | |
GFWYLCYLWSMJSC
|
8.3 | Kd | 3 | — | |
SCMPDMAJYNSKMW
|
8.3 | Kd | 3 | — | |
FIAJCYVGOYDLFU
|
8.2 | Kd | 3 | — | |
WPHKIQPVPYJNAX
|
8.2 | IC50 | 81 | — | |
UNGUWAMCUZJLAS
|
8.0 | Kd | 3 | — | |
HKSZLNNOFSGOKW
|
8.0 | Kd | 408 | — | |
KHDLZWDZNAKTKK
|
8.0 | Ki | 4 | Yes | |
ZJQWORQRPDYKRS
|
8.0 | Kd | 7 | — | |
CXQHYVUVSFXTMY
|
7.9 | Kd | 154 | — | |
LCVIRAZGMYMNNT
|
7.9 | IC50 | 4 | — | |
LCVIRAZGMYMNNT
|
7.9 | IC50 | 20 | — | |
SEJGTFPOEJWEGG
|
7.9 | Kd | 149 | — | |
QFOMGFNHXREHSV
|
7.9 | Kd | 3 | — | |
QKYQHNYADWTLSP
|
7.8 | Kd | 3 | — | |
FLBNLJLONKAPLR
|
7.8 | IC50 | 31 | — | |
YXMQIWJYPNBZJS
|
7.8 | IC50 | 4 | — | |
GBJVVSCPOBPEIT
|
7.8 | IC50 | 13 | Yes | |
LOGJQOUIVKBFGH
|
7.8 | IC50 | 11 | Yes | |
UFATYBRKMMRKGA
|
7.8 | Kd | 3 | — | |
FZTUPODAEPTYNG
|
7.7 | IC50 | 4 | Yes | |
JWILUIVAYLRFIY
|
7.7 | IC50 | 14 | — | |
HKSZLNNOFSGOKW
|
7.6 | Kd | 213 | — | |
HHFBDROWDBDFBR
|
7.6 | Kd | 40 | Yes | |
QQWUGDVOUVUTOY
|
7.5 | Kd | 231 | Yes | |
NHHQJBCNYHBUSI
|
7.4 | Kd | 220 | — | |
KGXBCWANASZZQG
|
7.3 | IC50 | 5 | — | |
YYLKKYCXAOBSRM
|
7.2 | Kd | 191 | — | |
ORWIYCURPDKSBI
|
7.2 | IC50 | 15 | Yes | |
XKFTZKGMDDZMJI
|
7.2 | IC50 | 64 | Yes | |
CPKWRHVMDOSXKE
|
7.2 | IC50 | 5 | — | |
LILXUVCZUBSSFA
|
7.2 | IC50 | 6 | — | |
MPVGZUGXCQEXTM
|
7.2 | Kd | 61 | Yes | |
LSEOXFVSQOHSDK
|
7.1 | Kd | 3 | — | |
KDKUVYLMPJIGKA
|
7.1 | Kd | 91 | Yes | |
MFWHDFGMXHATNR
|
6.9 | IC50 | 3 | — |