Target Details
| UniProt AC | Q9UQ88 |
|---|---|
| Gene Symbol | CDK11A |
| Protein Name | Cyclin-dependent kinase 11A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 26
- Clinical molecules 5
- Avg pChEMBL 6.61
Active Molecules (26)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WULUGQONDYDNKY
|
8.8 | IC50 | 5 | — | |
OVPNQJVDAFNBDN
|
8.3 | Kd | 44 | Yes | |
OUSFTKFNBAZUKL
|
7.3 | Kd | 58 | Yes | |
RAFISFVOOKCYLW
|
7.1 | IC50 | 6 | — | |
JWYHKDMZXSHNLA
|
7.0 | IC50 | 6 | — | |
KDKUVYLMPJIGKA
|
7.0 | Kd | 91 | Yes | |
LHMJTCJXGOQGEX
|
6.9 | IC50 | 6 | — | |
DQMDXHWHDMGPCC
|
6.8 | Kd | 6 | — | |
PUWXPMFEDYRLTM
|
6.7 | IC50 | 6 | — | |
GCIKSSRWRFVXBI
|
6.6 | Kd | 109 | Yes | |
CMJJZRAAQMUAFH
|
6.4 | Kd | 9 | — | |
PSPFQEBFYXJZEV
|
6.4 | Kd | 10 | — | |
WTDHONKZUZNMOZ
|
6.4 | IC50 | 6 | — | |
WIZPFVWZYLEGII
|
6.4 | IC50 | 6 | — | |
WMHURJYFLDPMEB
|
6.4 | Kd | 6 | — | |
KTEIFNKAUNYNJU
|
6.4 | Kd | 114 | — | |
CXQHYVUVSFXTMY
|
6.3 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
6.3 | Kd | 149 | — | |
VPDSZVYUHWYXCW
|
6.2 | IC50 | 6 | — | |
UISRWLSAXIOCND
|
6.2 | Kd | 5 | — | |
UXEWCQUEOJJYLF
|
6.0 | Kd | 6 | — | |
CHUDIJJINHPGKN
|
6.0 | IC50 | 6 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
QYZOGCMHVIGURT
|
6.0 | Kd | 26 | Yes |