Target Details
| UniProt AC | Q9UPZ9 |
|---|---|
| Gene Symbol | CILK1 |
| Protein Name | Serine/threonine-protein kinase ICK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 23
- Clinical molecules 8
- Avg pChEMBL 6.95
Associated Diseases (3)
Active Molecules (23)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BIIVYFLTOXDAOV
|
9.2 | Kd | 82 | Yes | |
JRNJNYBQQYBCLE
|
8.7 | Kd | 40 | Yes | |
XLSYZSRXVVCHLS
|
8.1 | Kd | 48 | — | |
OVPNQJVDAFNBDN
|
8.1 | Kd | 44 | Yes | |
MWKSRKSEWLRPBL
|
7.7 | Kd | 1075 | — | |
ZCCPLJOKGAACRT
|
7.5 | Kd | 599 | — | |
UIARLYUEJFELEN
|
7.4 | Kd | 289 | Yes | |
HKSZLNNOFSGOKW
|
7.4 | IC50 | 408 | — | |
UZWDCWONPYILKI
|
7.3 | Kd | 47 | — | |
OUSFTKFNBAZUKL
|
6.8 | Kd | 58 | Yes | |
AYCPARAPKDAOEN
|
6.6 | Kd | 73 | — | |
ZCBUQCWBWNUWSU
|
6.6 | Kd | 59 | — | |
HWXVIOGONBBTBY
|
6.6 | Kd | 27 | — | |
PIMQWRZWLQKKBJ
|
6.6 | Kd | 36 | — | |
OYONTEXKYJZFHA
|
6.4 | Kd | 69 | Yes | |
WINHZLLDWRZWRT
|
6.3 | Kd | 201 | Yes | |
BPNUQXPIQBZCMR
|
6.3 | Kd | 83 | Yes | |
AXRCEOKUDYDWLF
|
6.2 | Kd | 31 | — | |
MUOKSQABCJCOPU
|
6.0 | Kd | 36 | — | |
QLUYMIVVAYRECT
|
6.0 | Kd | 12 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |