Target Details
| UniProt AC | Q9UNQ0 |
|---|---|
| Gene Symbol | ABCG2 |
| Protein Name | Broad substrate specificity ATP-binding cassette transporter ABCG2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01061 (ABC2_membrane) PF19055 (ABC2_membrane_7) PF00005 (ABC_tran) |
Summary
- Multi-target molecules 52
- Clinical molecules 6
- Avg pChEMBL 6.7
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (52)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DWYRIWUZIJHQKQ
|
8.8 | IC50 | 3 | — | |
BQSJTQLCZDPROO
|
7.6 | IC50 | 3 | — | |
VOFLAIHEELWYGO
|
7.4 | IC50 | 2 | — | |
VNMQONKZFZQPCT
|
7.4 | IC50 | 3 | — | |
PHXJVRSECIGDHY
|
7.4 | IC50 | 59 | — | |
XPNBVAOZAHYCST
|
7.3 | IC50 | 3 | — | |
OEIXJPAIZADICN
|
7.3 | IC50 | 3 | — | |
GKDRMWXFWHEQQT
|
7.3 | IC50 | 7 | — | |
FCDNRJDHYPWDHC
|
7.2 | IC50 | 2 | — | |
SPMVMDHWKHCIDT
|
7.2 | IC50 | 30 | — | |
KQTJIUOOFLJRAY
|
7.1 | IC50 | 2 | — | |
CHAZSVOPUAINSR
|
7.1 | IC50 | 2 | — | |
HUILBFJFGUWXGF
|
7.1 | IC50 | 2 | — | |
KAZSKMJFUPEHHW
|
7.1 | IC50 | 2 | — | |
OEIXJPAIZADICN
|
7.0 | IC50 | 3 | — | |
AAKJLRGGTJKAMG
|
6.9 | IC50 | 50 | Yes | |
KBEUKMLEXDGSBY
|
6.9 | IC50 | 2 | — | |
PTVAOGIYBMTHSN
|
6.8 | IC50 | 2 | — | |
VZJNOIQBYQXEEZ
|
6.8 | IC50 | 2 | — | |
NRWKOPKPCJMFGI
|
6.8 | IC50 | 2 | — | |
FJHBVJOVLFPMQE
|
6.8 | IC50 | 2 | — | |
XPNBVAOZAHYCST
|
6.8 | IC50 | 3 | — | |
UBVZQGOVTLIHLH
|
6.7 | IC50 | 2 | — | |
BTYYWOYVBXILOJ
|
6.7 | IC50 | 4 | Yes | |
UHTHHESEBZOYNR
|
6.7 | IC50 | 66 | Yes | |
WHQCHUCQKNIQEC
|
6.7 | IC50 | 6 | — | |
VNMQONKZFZQPCT
|
6.7 | IC50 | 3 | — | |
YOURSKBAKQLDQW
|
6.7 | IC50 | 2 | — | |
OSFCMRGOZNQUSW
|
6.6 | IC50 | 2 | — | |
PJYWIMRIBDTXII
|
6.5 | IC50 | 2 | — | |
QKHVBGIOAYREBB
|
6.5 | IC50 | 2 | — | |
NECCTVFNAYKBCX
|
6.5 | IC50 | 3 | — | |
OTUOIHJJRAPDOB
|
6.4 | IC50 | 2 | — | |
ZPZDGGXNORFAFM
|
6.4 | IC50 | 4 | — | |
XGALLCVXEZPNRQ
|
6.3 | IC50 | 39 | Yes | |
IPXHDKAGTKPTNS
|
6.3 | IC50 | 2 | — | |
LVPXBXFMUREXPT
|
6.3 | IC50 | 2 | — | |
PMATZTZNYRCHOR
|
6.3 | Ki | 20 | — | |
RGLYKWWBQGJZGM
|
6.3 | IC50 | 8 | Yes | |
LGGHDPFKSSRQNS
|
6.3 | IC50 | 2 | — | |
HBGPQWXCRVPJIS
|
6.2 | IC50 | 2 | — | |
WMVUETDQMUIBJX
|
6.2 | IC50 | 2 | — | |
LCYPRFCDTJTQPG
|
6.2 | IC50 | 5 | — | |
KTUFNOKKBVMGRW
|
6.2 | IC50 | 38 | Yes | |
OIKGUIRGSMTFAP
|
6.2 | IC50 | 2 | — | |
JCKRZMGEVAGHHV
|
6.1 | IC50 | 2 | — | |
WSQDGWOFRGACTF
|
6.1 | IC50 | 2 | — | |
WKEBQZAUNGERGA
|
6.0 | IC50 | 2 | — | |
DTUCHVRTWHBOKV
|
6.0 | IC50 | 2 | — | |
VCOMYMMMFREKQC
|
6.0 | IC50 | 2 | — |