Target Details
| UniProt AC | Q9UNA0 |
|---|---|
| Gene Symbol | ADAMTS5 |
| Protein Name | A disintegrin and metalloproteinase with thrombospondin motifs 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17771 (ADAMTS_CR_2) PF19236 (ADAMTS_CR_3) PF05986 (ADAMTS_spacer1) PF01421 (Reprolysin) PF19030 (TSP1_ADAMTS) PF00090 (TSP_1) |
Summary
- Multi-target molecules 462
- Clinical molecules 24
- Avg pChEMBL 7.27
Active Molecules (462)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FVYLNTOUGPIPMM
|
6.6 | IC50 | 2 | — | |
VCENTKLGWWEJOU
|
6.6 | IC50 | 2 | — | |
ALDHNIAORPZUFG
|
6.5 | IC50 | 2 | — | |
SQGYSFDZVYSROA
|
6.5 | IC50 | 2 | — | |
ASVLCJFACSELPH
|
6.5 | IC50 | 2 | — | |
FCOHBGRTRWEGDQ
|
6.5 | IC50 | 2 | — | |
BOWBUENYNRWASZ
|
6.5 | IC50 | 2 | — | |
OGDMRINQXHOSNB
|
6.5 | IC50 | 2 | — | |
VNXAQUNXTGSDAD
|
6.5 | IC50 | 2 | — | |
JTPMXRVQNJQWPT
|
6.5 | IC50 | 2 | — | |
LSRFXDADRHAGGZ
|
6.5 | IC50 | 2 | — | |
ZMONONWLGUTMJN
|
6.5 | IC50 | 2 | — | |
RPHTYSCFXSHWBF
|
6.5 | IC50 | 2 | — | |
IENKEAFTWAFNOL
|
6.4 | IC50 | 2 | — | |
LSUCOXDOQAEXKL
|
6.4 | IC50 | 2 | — | |
VZJZHIKRRFMIGO
|
6.4 | IC50 | 2 | — | |
AABQMYBVWBDBKY
|
6.4 | IC50 | 2 | — | |
BHHZCJUKKKCRHQ
|
6.4 | IC50 | 2 | — | |
LBHGVAMLTISOJV
|
6.4 | IC50 | 2 | — | |
OUTUIYKUSHWASL
|
6.4 | IC50 | 2 | — | |
IMKDKHQDFFLOKK
|
6.4 | IC50 | 13 | Yes | |
NPBWCJCZUFCBEZ
|
6.4 | IC50 | 2 | — | |
BTKROMQYNIJXLC
|
6.3 | IC50 | 2 | — | |
QBZAPFWYAPXRGQ
|
6.3 | IC50 | 2 | — | |
KYGHQGXYBRYJIQ
|
6.3 | IC50 | 2 | — | |
LNIRXDCIYOBRPL
|
6.3 | IC50 | 3 | — | |
DDRRRYMVRWYNKI
|
6.3 | IC50 | 2 | — | |
YGEZZRWSTUOZOA
|
6.3 | IC50 | 2 | — | |
NITYDPDXAAFEIT
|
6.3 | IC50 | 20 | Yes | |
VYEJHVQIVKCLHC
|
6.3 | IC50 | 4 | Yes | |
YJRJYIQWWPZSTM
|
6.3 | IC50 | 6 | — | |
VFHNZPCBNRDGLE
|
6.3 | IC50 | 2 | — | |
HLLSMWRIVCVNPC
|
6.3 | IC50 | 2 | — | |
USQGYAOLZCMMRG
|
6.3 | IC50 | 2 | — | |
UKDQSIMWOVYUGX
|
6.2 | IC50 | 2 | — | |
IBSGSCYXBWXQDW
|
6.2 | IC50 | 4 | Yes | |
KYOXAYBXVWAPKV
|
6.2 | IC50 | 2 | — | |
CQARAIRTGMAYMZ
|
6.2 | Ki | 8 | — | |
NWFWLXVUCFLSOQ
|
6.2 | IC50 | 2 | — | |
OYVRPNKMOGLOSV
|
6.2 | IC50 | 2 | — | |
SGPBCFRSJZPAQO
|
6.2 | IC50 | 2 | — | |
ZVJILQAAQQNBOP
|
6.2 | IC50 | 6 | — | |
STVUCRKRBAWCPC
|
6.2 | IC50 | 4 | Yes | |
OWAWUDFSKQDLJG
|
6.2 | IC50 | 2 | — | |
LSPYJDKYIOCDAG
|
6.2 | IC50 | 2 | — | |
RJXBZPLCHUDNKA
|
6.2 | IC50 | 2 | — | |
QJGLVQUVXICDKT
|
6.2 | IC50 | 2 | — | |
GUEBRLZPFWEFBT
|
6.1 | IC50 | 2 | — | |
JHWOJEJVRYYQFM
|
6.1 | IC50 | 2 | — | |
YDMFQFGWICWKSM
|
6.1 | IC50 | 2 | — |