Target Details
| UniProt AC | Q9UNA0 |
|---|---|
| Gene Symbol | ADAMTS5 |
| Protein Name | A disintegrin and metalloproteinase with thrombospondin motifs 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17771 (ADAMTS_CR_2) PF19236 (ADAMTS_CR_3) PF05986 (ADAMTS_spacer1) PF01421 (Reprolysin) PF19030 (TSP1_ADAMTS) PF00090 (TSP_1) |
Summary
- Multi-target molecules 462
- Clinical molecules 24
- Avg pChEMBL 7.27
Active Molecules (462)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZMZUPFGBAXDKAM
|
6.9 | IC50 | 2 | — | |
DYWJWAJWDDNBGQ
|
6.9 | IC50 | 2 | — | |
FFTXPIXOKUHRLE
|
6.9 | IC50 | 2 | — | |
NVWYOERLHPCJLF
|
6.9 | IC50 | 2 | — | |
CXIDTYUJLXWEAY
|
6.9 | IC50 | 2 | — | |
IOOCYYNMZOYCGW
|
6.9 | IC50 | 2 | — | |
RAOQTAXXRGDVBS
|
6.9 | IC50 | 2 | — | |
QWGZIDLVLODPRW
|
6.8 | IC50 | 2 | — | |
BTIQTBAVWFZUGN
|
6.8 | IC50 | 2 | — | |
GPHYVVDMOPSOAK
|
6.8 | IC50 | 2 | — | |
MASAPOBQXDWROW
|
6.8 | IC50 | 2 | — | |
WRNVCIFWXDWAQY
|
6.8 | IC50 | 2 | — | |
CTRAVVYZOOTOPH
|
6.8 | IC50 | 2 | — | |
DXEOUZOCKYSZQC
|
6.8 | IC50 | 2 | — | |
MBFFAPVZPKHCKK
|
6.8 | IC50 | 2 | — | |
JRAYHZWPXHIVJI
|
6.8 | IC50 | 2 | — | |
OYVHTQLDQCPMLV
|
6.8 | IC50 | 2 | — | |
VVXZPLQFCWCGBS
|
6.8 | IC50 | 2 | — | |
KDRDHSZGYCDNRM
|
6.8 | IC50 | 2 | — | |
WAWUNJHTWVBKFW
|
6.8 | IC50 | 3 | — | |
YINSFKOGVSNIAY
|
6.8 | IC50 | 2 | — | |
RVYQNGRWJSISOS
|
6.8 | IC50 | 2 | — | |
XMWREONCCQNTDL
|
6.7 | IC50 | 2 | — | |
XZMNHVVTOKEKOE
|
6.7 | IC50 | 2 | — | |
ISXTYYPKYNPWCR
|
6.7 | IC50 | 2 | — | |
LOHKQXSWMQGIML
|
6.7 | IC50 | 2 | — | |
UMWZIHFBEHMTOZ
|
6.7 | IC50 | 2 | — | |
AFCXFUSGNPUIRN
|
6.7 | IC50 | 2 | — | |
SDZHRLYVISHMEO
|
6.7 | IC50 | 3 | — | |
RAAOGGVTKNNZQU
|
6.7 | IC50 | 2 | — | |
ZRAVABUPGXTUEH
|
6.7 | IC50 | 2 | — | |
FWVJBJBCMBAUIT
|
6.7 | IC50 | 2 | — | |
MWNUOLJFHXUUBS
|
6.7 | IC50 | 2 | — | |
FWVJBJBCMBAUIT
|
6.6 | IC50 | 2 | — | |
JRKDNBHZOWLDFD
|
6.6 | IC50 | 2 | — | |
MBVOSVDHUJIWRK
|
6.6 | IC50 | 2 | — | |
FFIKMUOIMXQHSI
|
6.6 | IC50 | 2 | — | |
FLTAYQGSMZKKCR
|
6.6 | IC50 | 2 | — | |
PSAIRTKPKUWNNP
|
6.6 | IC50 | 2 | — | |
MXNKXPGDSQYTQD
|
6.6 | IC50 | 2 | — | |
NZHFWSTVWWJDKQ
|
6.6 | IC50 | 2 | — | |
RLBVQFUDNZJYJM
|
6.6 | IC50 | 2 | — | |
STOLOTCLXZHFMA
|
6.6 | IC50 | 2 | — | |
HMVKTPIOGJURQF
|
6.6 | IC50 | 2 | — | |
LTNYDBXIBOIFNY
|
6.6 | IC50 | 2 | — | |
QIYIPIXAINLJLV
|
6.6 | IC50 | 2 | — | |
CSFRMTJLCGWESV
|
6.6 | IC50 | 2 | — | |
IIJIMCYNCLMHHL
|
6.6 | IC50 | 2 | — | |
IWRJDNKXMJBFEA
|
6.6 | IC50 | 2 | — | |
RVGJJKGKACPPHF
|
6.6 | IC50 | 2 | — |