Target Details
| UniProt AC | Q9UNA0 |
|---|---|
| Gene Symbol | ADAMTS5 |
| Protein Name | A disintegrin and metalloproteinase with thrombospondin motifs 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17771 (ADAMTS_CR_2) PF19236 (ADAMTS_CR_3) PF05986 (ADAMTS_spacer1) PF01421 (Reprolysin) PF19030 (TSP1_ADAMTS) PF00090 (TSP_1) |
Summary
- Multi-target molecules 462
- Clinical molecules 24
- Avg pChEMBL 7.27
Active Molecules (462)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZULTWIUGMFFCLD
|
7.2 | IC50 | 2 | — | |
IKHZGIGQISAUFN
|
7.2 | IC50 | 2 | — | |
VLNVWKDSFQRXHZ
|
7.2 | IC50 | 5 | Yes | |
CPYCKLJBTHKVRT
|
7.2 | IC50 | 3 | Yes | |
DYYJNBBMJXUGTR
|
7.2 | IC50 | 3 | — | |
KAWFVSYBDYABQU
|
7.2 | IC50 | 2 | — | |
ZGUHWFRFXRBHPL
|
7.2 | IC50 | 2 | — | |
QJBOHADGMLFYLD
|
7.2 | IC50 | 2 | — | |
NYSZVCQWENKRKM
|
7.2 | IC50 | 5 | Yes | |
REYQTRNKPUKDBL
|
7.2 | IC50 | 2 | — | |
GXCVJOQGIXISGY
|
7.2 | IC50 | 2 | — | |
ZKMBMHVMJIOBIH
|
7.2 | IC50 | 2 | — | |
SZEOXTMGYZKQHV
|
7.1 | IC50 | 4 | — | |
BBFYBNRNUNUHRO
|
7.1 | IC50 | 2 | — | |
BLPTVINPTQQNLV
|
7.1 | IC50 | 2 | — | |
CDVQKDXLTNVCDJ
|
7.1 | IC50 | 3 | — | |
CJYIEAVIAHNBAS
|
7.1 | IC50 | 2 | — | |
DBSGCGCAELIIMC
|
7.1 | IC50 | 2 | — | |
DNPHOKZQIKLZJT
|
7.1 | IC50 | 2 | — | |
DVMYRZMUQOTBGR
|
7.1 | IC50 | 2 | — | |
FUVOMTJFSKUMQI
|
7.1 | IC50 | 3 | — | |
FVGPYLWZRBWOTO
|
7.1 | IC50 | 2 | — | |
FWMBAODBFHUXLK
|
7.1 | IC50 | 2 | — | |
GLRLGVKPKCJBTN
|
7.1 | IC50 | 2 | — | |
HPZRYZXQQVTWJN
|
7.1 | IC50 | 3 | — | |
HVVNIZVKUPEBRS
|
7.1 | IC50 | 3 | — | |
JRFZSMAIBXKQOW
|
7.1 | IC50 | 3 | — | |
JTOKTYOQJGJDGG
|
7.1 | IC50 | 3 | — | |
KWDKDWAEPBDOBB
|
7.1 | IC50 | 2 | — | |
LBVBVIKJOWWVJX
|
7.1 | IC50 | 4 | — | |
LCPBZVLPMNYZLU
|
7.1 | IC50 | 2 | — | |
LQSHPJFKLZTHBV
|
7.1 | IC50 | 2 | — | |
LRTSAWNNQKOXFU
|
7.1 | IC50 | 2 | — | |
LVIZNCUABWKXTG
|
7.1 | IC50 | 3 | — | |
MGJMYLWAVDIBSV
|
7.1 | IC50 | 2 | — | |
NLNMKTSFGLFVDP
|
7.1 | IC50 | 2 | — | |
PTZGCAFYBLXVGN
|
7.1 | IC50 | 3 | — | |
QFSLYLOLLOXSPR
|
7.1 | IC50 | 3 | — | |
RAQSHADEFCYHMR
|
7.1 | IC50 | 2 | — | |
RPDOQOLWCQNQJE
|
7.1 | IC50 | 2 | — | |
RUAWTWDABHALSY
|
7.1 | IC50 | 3 | — | |
SZEIVIUBSTYPQJ
|
7.1 | IC50 | 2 | — | |
TZEBSVOXIIOOHD
|
7.1 | IC50 | 2 | — | |
UUIVHPQOLWYKFC
|
7.1 | IC50 | 3 | — | |
VHKRAQGLEXBWDL
|
7.1 | IC50 | 2 | — | |
XPUGDXRRGXHBML
|
7.1 | IC50 | 3 | — | |
XXQLCMDLJMBMLB
|
7.1 | IC50 | 3 | — | |
YDFSTSWRHBVFPJ
|
7.1 | IC50 | 2 | — | |
KXDVOTQQRPPFNY
|
7.1 | IC50 | 3 | — | |
BLPSVYQVAGCHMF
|
7.1 | IC50 | 2 | — |