Target Details
| UniProt AC | Q9UNA0 |
|---|---|
| Gene Symbol | ADAMTS5 |
| Protein Name | A disintegrin and metalloproteinase with thrombospondin motifs 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17771 (ADAMTS_CR_2) PF19236 (ADAMTS_CR_3) PF05986 (ADAMTS_spacer1) PF01421 (Reprolysin) PF19030 (TSP1_ADAMTS) PF00090 (TSP_1) |
Summary
- Multi-target molecules 462
- Clinical molecules 24
- Avg pChEMBL 7.27
Active Molecules (462)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KSLOIFYLMBDUDS
|
7.4 | IC50 | 2 | — | |
UDTINYVLJDOKAN
|
7.4 | IC50 | 3 | — | |
UJRBIZNZOPPPEC
|
7.4 | IC50 | 2 | — | |
XVMVNUAGECGGNK
|
7.4 | IC50 | 2 | — | |
ZPCSCHFHONOZPV
|
7.4 | IC50 | 2 | — | |
NPTUUUXCZCQNQS
|
7.4 | IC50 | 5 | — | |
ONOGZESTEFQIDC
|
7.4 | IC50 | 2 | — | |
WDAXMWCENYBRKO
|
7.4 | IC50 | 2 | — | |
HRHIVHWFCGOVGL
|
7.4 | IC50 | 2 | — | |
KFJVIDJSYPGQHH
|
7.4 | IC50 | 2 | — | |
HGVMZFIYNIXZLZ
|
7.3 | IC50 | 2 | — | |
MOWYZZPAPKVBEC
|
7.3 | IC50 | 2 | — | |
SYFMYEKYZWQZLV
|
7.3 | IC50 | 2 | — | |
WZHCTLSXWLCZEU
|
7.3 | IC50 | 2 | — | |
AFSFONATFSENCF
|
7.3 | IC50 | 2 | — | |
WECKJJDCDPVTTO
|
7.3 | IC50 | 3 | — | |
WRNVCIFWXDWAQY
|
7.3 | IC50 | 2 | — | |
HJGQFMIFDHXRQP
|
7.3 | IC50 | 2 | — | |
HTKFMVXDGZGNNW
|
7.3 | IC50 | 2 | — | |
INRSJNUJFBTCES
|
7.3 | IC50 | 2 | — | |
PWTMEJOXAUSTDY
|
7.3 | IC50 | 4 | — | |
RVGJJKGKACPPHF
|
7.3 | IC50 | 2 | — | |
ZMQVXCLMHVVMKI
|
7.3 | IC50 | 2 | — | |
KXUVWSDOPNGSBZ
|
7.3 | IC50 | 2 | — | |
OYCCHVFLJCOTKI
|
7.3 | IC50 | 2 | — | |
UOXSWFRPRZUDSH
|
7.3 | IC50 | 2 | — | |
VMRNKHLEOQDUMJ
|
7.3 | IC50 | 2 | — | |
CHTZMALPRVCUIK
|
7.3 | IC50 | 4 | — | |
HRZGFJYOHUVBRV
|
7.3 | IC50 | 2 | — | |
IABWDXKLHPEEBX
|
7.3 | IC50 | 2 | — | |
JDGHGRYBXRVLFH
|
7.3 | IC50 | 2 | — | |
QTWBSNWADUEERO
|
7.3 | IC50 | 2 | — | |
SOHSRXWNDMNQMJ
|
7.3 | IC50 | 2 | — | |
UUSOXZXTHXFMGV
|
7.3 | IC50 | 2 | — | |
UXTZIHLCCIDADG
|
7.3 | IC50 | 2 | — | |
VOANTRADBVMBCK
|
7.3 | IC50 | 2 | — | |
HRTBWTOXJOXCCB
|
7.3 | IC50 | 2 | — | |
MNKVQIVVYRSCJP
|
7.3 | IC50 | 2 | — | |
RZYRWVVQRWYGNG
|
7.3 | IC50 | 2 | — | |
CSFRMTJLCGWESV
|
7.2 | IC50 | 2 | — | |
FKHNOEWOJMNEPT
|
7.2 | IC50 | 2 | — | |
ROPVZXZEHJGNGB
|
7.2 | IC50 | 3 | — | |
CHBRRXABVNYHLG
|
7.2 | IC50 | 2 | — | |
MBFFAPVZPKHCKK
|
7.2 | IC50 | 2 | — | |
SXUFKFQWHMLFDQ
|
7.2 | IC50 | 2 | — | |
CBZOKXRPUYLLBY
|
7.2 | IC50 | 2 | — | |
RHLCNZXCMPRETL
|
7.2 | IC50 | 2 | — | |
DNZQEIOYACTIFD
|
7.2 | IC50 | 2 | — | |
KRFFMGOIPZCPLJ
|
7.2 | IC50 | 3 | — | |
XWUCDOCUSPAHFU
|
7.2 | IC50 | 2 | — |