Target Details
| UniProt AC | Q9UNA0 |
|---|---|
| Gene Symbol | ADAMTS5 |
| Protein Name | A disintegrin and metalloproteinase with thrombospondin motifs 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17771 (ADAMTS_CR_2) PF19236 (ADAMTS_CR_3) PF05986 (ADAMTS_spacer1) PF01421 (Reprolysin) PF19030 (TSP1_ADAMTS) PF00090 (TSP_1) |
Summary
- Multi-target molecules 462
- Clinical molecules 24
- Avg pChEMBL 7.27
Active Molecules (462)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DVWZDEQXQWWQOU
|
7.5 | IC50 | 3 | — | |
IJHSQTQFKJCKEA
|
7.5 | IC50 | 3 | — | |
USEQZALNBFQSDH
|
7.5 | IC50 | 3 | — | |
CHUAOQGPMXWHAQ
|
7.5 | IC50 | 2 | — | |
IHXLLQLBSUVNGK
|
7.5 | IC50 | 2 | — | |
MAQGKYQDMNIZTG
|
7.5 | IC50 | 2 | — | |
RCQCNSNJGRCTSZ
|
7.5 | IC50 | 3 | — | |
IYBHJPNFVKYDOX
|
7.5 | IC50 | 3 | — | |
LYUGBLDGSRTMRP
|
7.5 | IC50 | 2 | — | |
FWVMIBWFTPZCBI
|
7.5 | IC50 | 2 | — | |
JJVBXJPEBWHWEF
|
7.5 | IC50 | 2 | — | |
RWGLLJXXSHYVOK
|
7.5 | IC50 | 2 | — | |
RZKMGBZGSSSFLL
|
7.5 | IC50 | 2 | — | |
VJASAEQMGHZSFE
|
7.5 | IC50 | 2 | — | |
AONLPKICQLHFDZ
|
7.5 | IC50 | 2 | — | |
RSWPLKVUMZDBKI
|
7.5 | IC50 | 2 | — | |
DPKJSWSNGFNSEJ
|
7.4 | IC50 | 2 | — | |
AVLVMNPMCNZRPM
|
7.4 | IC50 | 3 | — | |
BBFYBNRNUNUHRO
|
7.4 | IC50 | 2 | — | |
BVFMJFRMGBKBIW
|
7.4 | IC50 | 3 | — | |
CRJZQBWHTWJUPJ
|
7.4 | IC50 | 3 | — | |
DLWUUXWPNZKTFO
|
7.4 | IC50 | 3 | — | |
FFYZDEBNTHTQDB
|
7.4 | IC50 | 3 | — | |
FSNZISYALYXUAH
|
7.4 | IC50 | 2 | — | |
FUENDAHGWXXXGO
|
7.4 | IC50 | 2 | — | |
GSBJFDQGAVFCLJ
|
7.4 | IC50 | 3 | — | |
IDQWSXMCWJZBFK
|
7.4 | IC50 | 3 | — | |
IUOVINQVOHJYDU
|
7.4 | IC50 | 3 | — | |
JSXIGTHUEBZKJY
|
7.4 | IC50 | 3 | — | |
LRTSAWNNQKOXFU
|
7.4 | IC50 | 3 | — | |
LTDJFOLMHATVKC
|
7.4 | IC50 | 3 | — | |
MARPMTNOLOIGKB
|
7.4 | IC50 | 2 | — | |
MJMKBSLUNYUWCO
|
7.4 | IC50 | 3 | — | |
MSDBLKCNXKEOHU
|
7.4 | IC50 | 3 | — | |
NAZJMGDZKSUZPA
|
7.4 | IC50 | 3 | — | |
QJQUJCFQIHPRTH
|
7.4 | IC50 | 2 | — | |
QJRMCRVDHSDQOQ
|
7.4 | IC50 | 3 | — | |
QKXZKYSXPIUZEA
|
7.4 | IC50 | 2 | — | |
RDAJPGITRGURGP
|
7.4 | IC50 | 3 | — | |
SVLANDCYAZJNPV
|
7.4 | IC50 | 3 | — | |
SZEIVIUBSTYPQJ
|
7.4 | IC50 | 2 | — | |
TZEBSVOXIIOOHD
|
7.4 | IC50 | 2 | — | |
UHWVEFMMEWDKEB
|
7.4 | IC50 | 2 | — | |
XZQFSKBVCGYHFA
|
7.4 | IC50 | 3 | — | |
YVHFKVFFSWECET
|
7.4 | IC50 | 2 | — | |
ANZVEJFIFVKQAS
|
7.4 | IC50 | 3 | — | |
WFFMEXQHWXEKBV
|
7.4 | IC50 | 2 | — | |
NVERRANKYVTEPN
|
7.4 | IC50 | 2 | — | |
ZLDUGCWRXAYWCQ
|
7.4 | IC50 | 2 | — | |
YGUZSRSJSPPSGU
|
7.4 | IC50 | 2 | — |