Target Details
| UniProt AC | Q9UNA0 |
|---|---|
| Gene Symbol | ADAMTS5 |
| Protein Name | A disintegrin and metalloproteinase with thrombospondin motifs 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17771 (ADAMTS_CR_2) PF19236 (ADAMTS_CR_3) PF05986 (ADAMTS_spacer1) PF01421 (Reprolysin) PF19030 (TSP1_ADAMTS) PF00090 (TSP_1) |
Summary
- Multi-target molecules 462
- Clinical molecules 24
- Avg pChEMBL 7.27
Active Molecules (462)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HNYCVJJYDZYSOS
|
7.7 | IC50 | 2 | — | |
JDBUKSMCZPXYJU
|
7.7 | IC50 | 4 | — | |
QMEYEEICXNLCJY
|
7.7 | IC50 | 2 | — | |
RZRHUPMJEFKEEG
|
7.7 | IC50 | 2 | — | |
SIXCEPSXNLUZTE
|
7.7 | IC50 | 2 | — | |
AHXGZLJBINZPQZ
|
7.7 | IC50 | 3 | Yes | |
ASLMJZFVIFDYPI
|
7.7 | IC50 | 2 | — | |
KNNZSFMCVFUPON
|
7.7 | IC50 | 2 | — | |
MAQGKYQDMNIZTG
|
7.7 | IC50 | 2 | — | |
OTCWHHBFFQOWCU
|
7.7 | IC50 | 2 | — | |
NVCCYYKMLFBFPP
|
7.7 | IC50 | 3 | — | |
QMEYEEICXNLCJY
|
7.7 | IC50 | 2 | — | |
AFUQYGWPKAMIBT
|
7.7 | IC50 | 2 | — | |
JFUFPMIABSBLEE
|
7.7 | IC50 | 2 | — | |
KTSVBNSBXWVDTE
|
7.7 | IC50 | 3 | — | |
OBQNFIXICFYDBT
|
7.7 | IC50 | 3 | — | |
OJISSJZEUBCVQI
|
7.7 | IC50 | 2 | — | |
QRKXZIVWYBYWEG
|
7.7 | IC50 | 2 | — | |
XODHZTSNMPEPED
|
7.7 | IC50 | 2 | — | |
XUGGLUHGDWIBGT
|
7.7 | IC50 | 2 | — | |
KFOJCCXBEQXGOL
|
7.6 | IC50 | 3 | Yes | |
LLZNOGUPMFYFGU
|
7.6 | IC50 | 3 | — | |
QMEYEEICXNLCJY
|
7.6 | IC50 | 2 | — | |
UAGAABCJKYADIR
|
7.6 | IC50 | 3 | — | |
BMAHWOMMEYMRNY
|
7.6 | IC50 | 2 | — | |
UUNGDQWYHHDBHV
|
7.6 | IC50 | 2 | — | |
XUAZQANALKLDEW
|
7.6 | IC50 | 2 | — | |
YLSHULIHKQRKEM
|
7.6 | IC50 | 4 | — | |
HYOFXPHIEQTJFW
|
7.6 | IC50 | 2 | — | |
OACIIQIUQKQGAD
|
7.6 | IC50 | 2 | — | |
ONWZTEISEVDFER
|
7.6 | IC50 | 2 | — | |
RSWPLKVUMZDBKI
|
7.6 | IC50 | 2 | — | |
NGADEBBDUSTEJD
|
7.6 | IC50 | 2 | — | |
MKGHITYLXXYNMZ
|
7.6 | IC50 | 3 | — | |
NPWGFJCNOCYDSO
|
7.6 | IC50 | 2 | — | |
QRHNXIGPFHVEIB
|
7.6 | IC50 | 2 | — | |
SSXHPSBZPUTJCO
|
7.6 | IC50 | 3 | — | |
QVLRRQHYUCZYFV
|
7.6 | IC50 | 3 | — | |
UURCCWSAXNITTQ
|
7.6 | IC50 | 2 | — | |
SPAODDWHKVLWKW
|
7.6 | IC50 | 2 | — | |
IXVRORAFKAVRDP
|
7.5 | IC50 | 2 | — | |
QQCNGNFIZAKQDT
|
7.5 | IC50 | 4 | — | |
XDCORYPKECEONK
|
7.5 | IC50 | 2 | — | |
HHHJVFVJVOPDRT
|
7.5 | IC50 | 3 | — | |
QVFLVOHFXMNIFB
|
7.5 | IC50 | 3 | Yes | |
CCYLLSFOUYRFAH
|
7.5 | IC50 | 2 | — | |
JSHMJRSKCZIJHA
|
7.5 | IC50 | 2 | — | |
KNKPUUINTPWUPH
|
7.5 | IC50 | 3 | — | |
WRNVCIFWXDWAQY
|
7.5 | IC50 | 2 | — | |
ZAZABNIPHQNPKB
|
7.5 | IC50 | 2 | — |