Target Details
| UniProt AC | Q9UNA0 |
|---|---|
| Gene Symbol | ADAMTS5 |
| Protein Name | A disintegrin and metalloproteinase with thrombospondin motifs 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17771 (ADAMTS_CR_2) PF19236 (ADAMTS_CR_3) PF05986 (ADAMTS_spacer1) PF01421 (Reprolysin) PF19030 (TSP1_ADAMTS) PF00090 (TSP_1) |
Summary
- Multi-target molecules 462
- Clinical molecules 24
- Avg pChEMBL 7.27
Active Molecules (462)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LDIAENRSEDNGCJ
|
7.9 | IC50 | 2 | — | |
ABNKQEYPWPPOOQ
|
7.9 | IC50 | 3 | — | |
BEYBREWPWQEWSI
|
7.9 | IC50 | 3 | — | |
CVXZBZOHZGZICE
|
7.9 | IC50 | 3 | — | |
FWMBAODBFHUXLK
|
7.9 | IC50 | 2 | — | |
HBRVHODOXCBKHN
|
7.9 | IC50 | 3 | — | |
IHRJQBVRWWFMFZ
|
7.9 | IC50 | 3 | — | |
JSUBEBYUGKGELF
|
7.9 | IC50 | 3 | — | |
KQDWIZNOSHZMAC
|
7.9 | IC50 | 3 | — | |
LBEBGRPTXSMXMO
|
7.9 | IC50 | 3 | — | |
MDCDJAYEONMPDM
|
7.9 | IC50 | 3 | — | |
MDCDJAYEONMPDM
|
7.9 | IC50 | 3 | — | |
RDWFDWWQRNYJGA
|
7.9 | IC50 | 3 | — | |
RKELHXSYFGUUBO
|
7.9 | IC50 | 3 | — | |
VUBCFWBRGYOPKR
|
7.9 | IC50 | 3 | — | |
ZEMLAXHMFOILNW
|
7.9 | IC50 | 3 | — | |
YGTSAUDEZYDSGM
|
7.9 | IC50 | 2 | — | |
VJASAEQMGHZSFE
|
7.9 | IC50 | 2 | — | |
PKTAGMTUNRVAKO
|
7.9 | IC50 | 2 | — | |
UOXSWFRPRZUDSH
|
7.9 | IC50 | 2 | — | |
KISNQJUMQDMWMF
|
7.8 | IC50 | 3 | — | |
MKGHITYLXXYNMZ
|
7.8 | IC50 | 3 | — | |
LBFZDWQGADLLKS
|
7.8 | IC50 | 2 | — | |
DLWHWYIHKZASJX
|
7.8 | IC50 | 2 | — | |
SFQHPECSYRCUKU
|
7.8 | IC50 | 2 | — | |
YILYUDCSMINQHO
|
7.8 | IC50 | 3 | — | |
ZRQWUQCXSKEXGA
|
7.8 | Ki | 6 | — | |
UKSOPPJLMFZIFG
|
7.8 | IC50 | 2 | — | |
QRNZXNUHQIYSQV
|
7.8 | IC50 | 2 | — | |
XUOKZLGAMXUMSE
|
7.8 | IC50 | 3 | — | |
ZQBRQDVCSATBBO
|
7.8 | IC50 | 2 | — | |
LDDKAYGLGQWILO
|
7.8 | IC50 | 6 | — | |
CVBUIFHDZMEAIE
|
7.8 | IC50 | 2 | — | |
XTTXOVQPTVWBOC
|
7.8 | IC50 | 2 | — | |
DSLRBIQFKOUGKT
|
7.8 | IC50 | 4 | Yes | |
FCEJLOVSBUDTHL
|
7.8 | IC50 | 2 | — | |
KHOCDFJBVDAQHO
|
7.8 | IC50 | 2 | — | |
UACUZULRKJKTHE
|
7.8 | IC50 | 5 | Yes | |
HYCYFNRXRRBATO
|
7.8 | IC50 | 3 | — | |
LHERXAOZMZIVQX
|
7.8 | IC50 | 2 | — | |
INOYENJSYPDBEC
|
7.8 | IC50 | 3 | — | |
LHKXLEZLEFHFJV
|
7.7 | IC50 | 3 | — | |
MNUPPLNWLDYAPV
|
7.7 | IC50 | 2 | — | |
ARVDGBFKIFLARF
|
7.7 | IC50 | 3 | — | |
OJPRZTDTKMGAMY
|
7.7 | IC50 | 3 | Yes | |
UHKJKGYIHRIXMQ
|
7.7 | IC50 | 2 | — | |
UOXSWFRPRZUDSH
|
7.7 | IC50 | 2 | — | |
WIKRDIGSYVQGTH
|
7.7 | IC50 | 2 | — | |
ZIXRMLDHKPIARA
|
7.7 | IC50 | 3 | — | |
CMLVKUWQFZQPPS
|
7.7 | IC50 | 3 | — |