Target Details
| UniProt AC | Q9UNA0 |
|---|---|
| Gene Symbol | ADAMTS5 |
| Protein Name | A disintegrin and metalloproteinase with thrombospondin motifs 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17771 (ADAMTS_CR_2) PF19236 (ADAMTS_CR_3) PF05986 (ADAMTS_spacer1) PF01421 (Reprolysin) PF19030 (TSP1_ADAMTS) PF00090 (TSP_1) |
Summary
- Multi-target molecules 462
- Clinical molecules 24
- Avg pChEMBL 7.27
Active Molecules (462)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CAFLLFZUWQCIHM
|
6.1 | IC50 | 2 | — | |
GSHKFLCNIDFHJZ
|
6.1 | IC50 | 2 | — | |
ISHINUUQDKDNHQ
|
6.1 | IC50 | 2 | — | |
ADDJDJQFPKUMAF
|
6.1 | Ki | 7 | — | |
IOBCRLWDQPOVFD
|
6.1 | IC50 | 2 | — | |
CTWWCYYGTKSRCU
|
6.0 | IC50 | 2 | — | |
FFCQFLOKIRUZOS
|
6.0 | IC50 | 3 | — | |
RVJWHYWBFQXTCP
|
6.0 | IC50 | 2 | — | |
AUSYXXOLFARXLL
|
6.0 | IC50 | 2 | — | |
BZUGNOPIQMYMFU
|
6.0 | IC50 | 2 | — | |
PGVYYPZKXKGBLD
|
6.0 | Ki | 2 | — | |
VPPAFDVKUDHCGQ
|
6.0 | IC50 | 2 | — |