Target Details
| UniProt AC | Q9UNA0 |
|---|---|
| Gene Symbol | ADAMTS5 |
| Protein Name | A disintegrin and metalloproteinase with thrombospondin motifs 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17771 (ADAMTS_CR_2) PF19236 (ADAMTS_CR_3) PF05986 (ADAMTS_spacer1) PF01421 (Reprolysin) PF19030 (TSP1_ADAMTS) PF00090 (TSP_1) |
Summary
- Multi-target molecules 462
- Clinical molecules 24
- Avg pChEMBL 7.27
Active Molecules (462)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FTEPMVFWUZEGMB
|
9.7 | IC50 | 2 | — | |
NPTUUUXCZCQNQS
|
9.0 | IC50 | 4 | — | |
GBGAKFWYCGVPHY
|
8.8 | IC50 | 7 | Yes | |
BWKAHABETZLDBG
|
8.8 | IC50 | 2 | — | |
OHLDJJXRTLZQSU
|
8.7 | IC50 | 3 | — | |
JHOUEQAOHDTLPY
|
8.7 | IC50 | 4 | — | |
VCOUEHUEFUDZIS
|
8.7 | IC50 | 2 | — | |
XTJBTJMEXZEGIF
|
8.7 | IC50 | 6 | — | |
HBHHQROCMYJFKL
|
8.7 | IC50 | 2 | — | |
NKLVBHMAIMEVEH
|
8.6 | IC50 | 2 | — | |
SGSKDJMEPQTYQW
|
8.6 | IC50 | 2 | — | |
DNSIVPJNRUSHDP
|
8.5 | IC50 | 4 | Yes | |
DAWHPQGJJMGZKV
|
8.5 | Ki | 2 | — | |
PLZHEWIMJLHYQI
|
8.5 | Ki | 2 | — | |
GNFWJCGIZJCASB
|
8.4 | IC50 | 2 | — | |
BXOAWISKNWMSMA
|
8.4 | IC50 | 2 | — | |
IHWBLYROWNAFFC
|
8.4 | IC50 | 2 | — | |
VXEBTZZUKSNQHZ
|
8.4 | IC50 | 2 | — | |
AEVUQVQJMYYUSL
|
8.4 | IC50 | 2 | — | |
FJEJHTFPLBTMLO
|
8.4 | IC50 | 4 | — | |
ASSAXYGADPLJMQ
|
8.4 | IC50 | 2 | — | |
BNJKWXPRZSOHBL
|
8.3 | IC50 | 2 | — | |
CHUAOQGPMXWHAQ
|
8.3 | IC50 | 2 | — | |
LKGCROMJAWADLL
|
8.3 | IC50 | 2 | — | |
ZPUWHZPEHISDSA
|
8.3 | IC50 | 2 | — | |
MYNRCIAHZNZKOZ
|
8.2 | Ki | 2 | — | |
LTVIJEFEZVFIST
|
8.2 | IC50 | 14 | Yes | |
GYAIYJXOPICREB
|
8.2 | IC50 | 2 | — | |
LDIAENRSEDNGCJ
|
8.2 | IC50 | 2 | — | |
GRSFKJZRDUZQPW
|
8.1 | IC50 | 9 | Yes | |
RWUSOKGVCNRFRC
|
8.1 | IC50 | 2 | — | |
OHLDJJXRTLZQSU
|
8.1 | IC50 | 2 | — | |
RDRCRROFSMSFED
|
8.1 | IC50 | 2 | — | |
VXXYNKXMRXANKX
|
8.1 | IC50 | 2 | — | |
PENUDEJHXUSMIL
|
8.1 | IC50 | 4 | Yes | |
RDRCRROFSMSFED
|
8.1 | IC50 | 2 | — | |
KIMAXDZENSBFAC
|
8.1 | IC50 | 3 | Yes | |
JHBAOENFEKRBLY
|
8.1 | Ki | 2 | — | |
VJASAEQMGHZSFE
|
8.1 | IC50 | 2 | — | |
FTPFWQRREQUXLQ
|
8.0 | IC50 | 3 | Yes | |
GYSTVJYXBPSVIF
|
8.0 | Ki | 4 | — | |
OVPSSIXIRKPDEH
|
8.0 | IC50 | 2 | — | |
FHIRATRLDJRXHH
|
8.0 | IC50 | 2 | — | |
KXFPWCKTSXRQIS
|
8.0 | IC50 | 4 | — | |
OOQSIBQKXZCHOC
|
8.0 | IC50 | 3 | — | |
VKMTZVHITCDFFV
|
8.0 | IC50 | 2 | — | |
PDBQNZHFRVAZBC
|
7.9 | IC50 | 2 | — | |
LBFZDWQGADLLKS
|
7.9 | IC50 | 2 | — | |
RKYYWBHSYPIJKC
|
7.9 | IC50 | 4 | — | |
VAKWUGCSPIRJRO
|
7.9 | IC50 | 3 | — |