Target Details
UniProt ACQ9UN88
Gene SymbolGABRQ
Protein NameGamma-aminobutyric acid receptor subunit theta
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 325
  • Clinical molecules 0
  • Avg pChEMBL 7.41
Top Co-occurrence Targets
Active Molecules (325)
InChIKey pChEMBL Type Targets Clinical
CELFESKDAXZKDL 6.6 IC50 16
HXXGVDKGNHCARX 6.6 IC50 16
VMNYVCMDPUOQEL 6.6 Ki 16
GXFWOMYQHNODFA 6.6 IC50 16
HOTHDLMXYUFPSZ 6.6 IC50 16
QQONDVXXMVPYIB 6.6 Ki 16
GCNSLTKPBZQFJK 6.6 IC50 16
ODIZUHKZJZYZAL 6.6 IC50 16
RTMFRAUTYIKCRK 6.6 Ki 16
WNDIDYSCZWXEJF 6.6 Ki 16
LOBNIVNGRUTMOS 6.5 IC50 16
WRUTXEAYYQYJHO 6.5 Ki 16
HJGRBNHROFTASJ 6.5 IC50 16
YHZXFRGWTKYPKS 6.5 Ki 16
GAQCKHAXURZXGX 6.5 IC50 16
VEWLYIAEUXDQBW 6.5 IC50 16
GDVGLPNNOCDLLD 6.5 IC50 16
GEFDSAOHFGLQEZ 6.5 Ki 17
WCTCMHZWHMFZFN 6.5 Ki 17
DDSULWHSYUPHBK 6.5 IC50 16
XRWYYMUIIXMQBL 6.5 IC50 16
DAYQXLQRTQODQF 6.4 Ki 16
DNCFKDLZZSXXJP 6.4 IC50 16
MUPIUJYENVWEKT 6.4 IC50 16
NQFQEBQBZXSXIX 6.4 IC50 16
VNFZCRPFALLSNM 6.4 IC50 16
SQPWTARSPNZNEI 6.4 IC50 16
QCSFXCHHKYXLHE 6.4 Ki 16
YFEZLTPSCJWVHI 6.4 Ki 16
YOJAHANNNITYMX 6.4 Ki 16
ZLAPTIDQRXJQQL 6.4 IC50 16
AEPFXRGRJZMVIF 6.3 Ki 17
JBTLCAMUYYCXTA 6.3 IC50 16
DKCNNHVHQYMVTO 6.3 IC50 16
BDGWCPYUERFMMY 6.3 Ki 16
UMYWGMKUCZAQJO 6.3 Ki 16
FNZFELZOBRBQJY 6.3 IC50 16
IGCSLIVTBUKKRS 6.3 IC50 16
SRJOCJYGOFTFLH 6.3 Ki 16
IKDYRDIWKFJQTR 6.3 IC50 16
PZWMQJZDDYQYGN 6.3 Ki 16
ZEEOGWVZWOURAE 6.2 Ki 16
OMGOVFIKWLKTPS 6.2 Ki 16
BZIBRALMCDHACX 6.2 Ki 17
JWTQJUQJIRWZLA 6.2 Ki 16
ODWCGGCCGLKRAK 6.2 Ki 16
ICRYUJPBYIPXQF 6.2 IC50 16
ZMKDYQONTIIETL 6.2 Ki 16
OJOTYQLMNVPQBO 6.2 Ki 16
RRAXPPHKWFOGGL 6.2 Ki 16
2D structure