Target Details
| UniProt AC | Q9UN88 |
|---|---|
| Gene Symbol | GABRQ |
| Protein Name | Gamma-aminobutyric acid receptor subunit theta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 325
- Clinical molecules 0
- Avg pChEMBL 7.41
KEGG Pathways (7)
Active Molecules (325)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CKZVPJOTELQSHC
|
7.8 | IC50 | 16 | — | |
QCHBQARHFYCDNV
|
7.8 | IC50 | 16 | — | |
ZFPVOBQMGRHOBJ
|
7.8 | IC50 | 16 | — | |
JWZNKJCEYMWLHS
|
7.8 | IC50 | 16 | — | |
MEWGBPFYMUBENF
|
7.8 | IC50 | 16 | — | |
NAXZRUMPHRMRDF
|
7.8 | IC50 | 16 | — | |
VXOXRIDQOBACKW
|
7.8 | Ki | 16 | — | |
YJYRFBZSNPRHKU
|
7.8 | IC50 | 16 | — | |
QVBUOPGWPXUAHT
|
7.7 | IC50 | 16 | — | |
UIPGLQFPZVUUQW
|
7.7 | Ki | 16 | — | |
VQENDYBPFSSMNH
|
7.7 | IC50 | 16 | — | |
BYEKIJACVDAPTD
|
7.7 | Ki | 16 | — | |
LLAKESJIQFAQJA
|
7.7 | IC50 | 16 | — | |
FQDQLHDSVITISC
|
7.7 | IC50 | 16 | — | |
HKLYPSSDHPAOJM
|
7.7 | IC50 | 16 | — | |
RSEMKXACIMVTQP
|
7.7 | Ki | 16 | — | |
WRDHNUVAWMYMJK
|
7.7 | IC50 | 16 | — | |
AURFZBICLPNKBZ
|
7.7 | IC50 | 16 | — | |
ZFLBRINMIQTFNB
|
7.7 | Ki | 18 | — | |
CJYPUCKDMBCYEH
|
7.6 | IC50 | 16 | — | |
LNPSYDJGQQETLB
|
7.6 | Ki | 16 | — | |
SHTOUNSWZVCSOU
|
7.6 | IC50 | 16 | — | |
TWQDMCPDTPVCQP
|
7.6 | IC50 | 16 | — | |
VHQCVUYEMJHQEX
|
7.6 | Ki | 16 | — | |
JHDNCJGODWCHES
|
7.6 | IC50 | 16 | — | |
LIXHLXZPUZQKCT
|
7.6 | IC50 | 16 | — | |
MBBOXTKOOFAZLI
|
7.6 | IC50 | 16 | — | |
PDOZRVXKPBQAJH
|
7.6 | IC50 | 16 | — | |
JWLCOGXPTWMMDY
|
7.6 | Ki | 16 | — | |
KBVJZOBCOIANOX
|
7.6 | Ki | 16 | — | |
KOMBGWPXIHBMLL
|
7.6 | IC50 | 16 | — | |
OSHQANHMWJQRHB
|
7.6 | Ki | 16 | — | |
ULMKSNRBNFFOJQ
|
7.6 | Ki | 16 | — | |
ZWJGDMSWCKASII
|
7.6 | IC50 | 16 | — | |
HSUCRXNJMPDNOG
|
7.6 | IC50 | 16 | — | |
JNWDOTPNEZYWGO
|
7.6 | Ki | 16 | — | |
JAFQEKAQGSQGTM
|
7.6 | Ki | 16 | — | |
KQTMWRZAVOUNCI
|
7.6 | IC50 | 16 | — | |
VIEKPLVJCPXIIB
|
7.6 | IC50 | 16 | — | |
XLKKKDPUVUIHEL
|
7.6 | IC50 | 16 | — | |
AANJEGNNNSDLGW
|
7.5 | Ki | 16 | — | |
WPJDKKSDGLIQQB
|
7.5 | Ki | 16 | — | |
DRCGHGOPCPUYAI
|
7.5 | IC50 | 16 | — | |
NKIYALPHXLYICR
|
7.5 | IC50 | 16 | — | |
BTCSSZJGUNDROE
|
7.5 | Ki | 23 | — | |
FOSOKBNWILBLSN
|
7.5 | Ki | 16 | — | |
KTFRBKXLNKKPEA
|
7.5 | IC50 | 16 | — | |
ACVGNKYJVGNLIL
|
7.5 | IC50 | 16 | — | |
SCAPGUIFNHZJLH
|
7.5 | IC50 | 16 | — | |
SUONVKFDJJYYME
|
7.5 | IC50 | 16 | — |